| 1 |
33610566 | Potential Determinants for Metabolic Fates and Inhibitory Effects of Isobavachalcone Involving in Human Cytochrome P450, UDP-Glucuronosyltransferase Enzymes, and Efflux Transporters. | 2021 May |
1 |
| 2 |
34133540 | Association of UGT1A6 gene polymorphism with clinical outcome in pediatric epileptic patients on sodium valproate monotherapy. | 2021 |
1 |
| 3 |
34192355 | Inhibition of human UDP-glucuronosyltransferase enzyme by Dabrafenib: Implications for drug-drug interactions. | 2021 Nov |
2 |
| 4 |
33008919 | Arginine-259 of UGT2B7 Confers UDP-Sugar Selectivity. | 2020 Dec |
1 |
| 5 |
31163218 | S-equol glucuronidation in liver and intestinal microsomes of humans, monkeys, dogs, rats, and mice. | 2019 Sep |
2 |
| 6 |
27405656 | Glucuronidation of 4-tert-octylphenol in humans, monkeys, rats, and mice: an in vitro analysis using liver and intestine microsomes. | 2017 Mar |
2 |
| 7 |
28266877 | Glucuronidation: driving factors and their impact on glucuronide disposition. | 2017 May |
4 |
| 8 |
28500425 | Hepatic glucuronidation of 4-tert-octylphenol in humans: inter-individual variability and responsible UDP-glucuronosyltransferase isoforms. | 2017 Nov |
2 |
| 9 |
26514348 | Hepatic and intestinal glucuronidation of mono(2-ethylhexyl) phthalate, an active metabolite of di(2-ethylhexyl) phthalate, in humans, dogs, rats, and mice: an in vitro analysis using microsomal fractions. | 2016 Jul |
2 |
| 10 |
25034008 | Glucuronidation of fimasartan, a new angiotensin receptor antagonist, is mainly mediated by UGT1A3. | 2015 Jan |
1 |
| 11 |
25684194 | Inhibition screening method of microsomal UGTs using the cocktail approach. | 2015 Apr 25 |
1 |
| 12 |
23888985 | Comparing the glucuronidation capacity of the feline liver with substrate-specific glucuronidation in dogs. | 2014 Feb |
1 |
| 13 |
24854283 | In vitro glucuronidation of five rhubarb anthraquinones by intestinal and liver microsomes from humans and rats. | 2014 Aug 5 |
1 |
| 14 |
23277092 | Variability in UDP-glucuronosyltransferase genes and morphine metabolism: observations from a cross-sectional multicenter study in advanced cancer patients with pain. | 2013 Mar |
2 |
| 15 |
23362992 | Identification of flavone glucuronide isomers by metal complexation and tandem mass spectrometry: regioselectivity of uridine 5'-diphosphate-glucuronosyltransferase isozymes in the biotransformation of flavones. | 2013 Feb 20 |
1 |
| 16 |
22050083 | Quantification of human uridine-diphosphate glucuronosyl transferase 1A isoforms in liver, intestine, and kidney using nanobore liquid chromatography-tandem mass spectrometry. | 2012 Jan 3 |
2 |
| 17 |
22071170 | UDP-glucuronosyltransferase (UGT) 1A9-overexpressing HeLa cells is an appropriate tool to delineate the kinetic interplay between breast cancer resistance protein (BRCP) and UGT and to rapidly identify the glucuronide substrates of BCRP. | 2012 Feb |
1 |
| 18 |
22814440 | Stereoselective glucuronidation of carvedilol in human liver and intestinal microsomes. | 2012 |
2 |
| 19 |
22982073 | Coupling of UDP-glucuronosyltransferases and multidrug resistance-associated proteins is responsible for the intestinal disposition and poor bioavailability of emodin. | 2012 Dec 15 |
1 |
| 20 |
21622626 | Sequential metabolism of sesamin by cytochrome P450 and UDP-glucuronosyltransferase in human liver. | 2011 Sep |
1 |
| 21 |
21937736 | Raloxifene glucuronidation in human intestine, kidney, and liver microsomes and in human liver microsomes genotyped for the UGT1A1*28 polymorphism. | 2011 Dec |
2 |
| 22 |
20713656 | Metabolism of 1'- and 4-hydroxymidazolam by glucuronide conjugation is largely mediated by UDP-glucuronosyltransferases 1A4, 2B4, and 2B7. | 2010 Nov |
1 |
| 23 |
21175442 | Repaglinide-gemfibrozil drug interaction: inhibition of repaglinide glucuronidation as a potential additional contributing mechanism. | 2010 Dec |
1 |
| 24 |
17991766 | Resveratrol (trans-resveratrol, 3,5,4'-trihydroxy-trans-stilbene) glucuronidation exhibits atypical enzyme kinetics in various protein sources. | 2008 Feb |
1 |
| 25 |
18537579 | Liver-enriched transcription factors and their role in regulating UDP glucuronosyltransferase gene expression. | 2008 Jun |
1 |
| 26 |
17446261 | Predominant contribution of UDP-glucuronosyltransferase 2B7 in the glucuronidation of racemic flurbiprofen in the human liver. | 2007 Jul |
1 |
| 27 |
16518089 | [Pharmacokinetics and disposition of silodosin (KMD-3213)]. | 2006 Mar |
1 |
| 28 |
16595710 | Human UDP-glucuronosyltransferase, UGT1A8, glucuronidates dihydrotestosterone to a monoglucuronide and further to a structurally novel diglucuronide. | 2006 Jul |
2 |
| 29 |
16887906 | Isoform-specific regulation of uridine diphosphate-glucuronosyltransferase 2B enzymes in the human prostate: differential consequences for androgen and bioactive lipid inactivation. | 2006 Nov |
2 |
| 30 |
15845768 | Phosphorylation of a UDP-glucuronosyltransferase regulates substrate specificity. | 2005 May 3 |
1 |
| 31 |
14744950 | Identification of human UDP-glucuronosyltransferase enzyme(s) responsible for the glucuronidation of posaconazole (Noxafil). | 2004 Feb |
2 |
| 32 |
15304429 | Drug-drug interactions for UDP-glucuronosyltransferase substrates: a pharmacokinetic explanation for typically observed low exposure (AUCi/AUC) ratios. | 2004 Nov |
1 |
| 33 |
15535854 | Metabolic inactivation of estrogens in breast tissue by UDP-glucuronosyltransferase enzymes: an overview. | 2004 |
1 |
| 34 |
12639971 | Glucuronidation of arachidonic and linoleic acid metabolites by human UDP-glucuronosyltransferases. | 2003 Jun |
1 |
| 35 |
11316519 | Natural and synthetic inhibitors of UDP-glucuronosyltransferase. | 2001 Feb |
1 |
| 36 |
11355849 | High-performance liquid chromatographic method combining radiochemical and ultraviolet detection for determination of low activities of uridine 5'-diphosphate-glucuronosyltransferase. | 2001 May 15 |
1 |
| 37 |
11038168 | The specificity of glucuronidation of entacapone and tolcapone by recombinant human UDP-glucuronosyltransferases. | 2000 Nov |
1 |
| 38 |
11134149 | Cellular localization of uridine diphosphoglucuronosyltransferase 2B enzymes in the human prostate by in situ hybridization and immunohistochemistry. | 2000 Dec |
2 |
| 39 |
9895303 | Cloning and characterization of a simian UDP-glucuronosyltransferase enzyme UGT2B20, a novel C19 steroid-conjugating protein. | 1999 Feb 1 |
1 |
| 40 |
9406655 | Structure and function of uridine diphosphate glucuronosyltransferases. | 1997 Dec |
1 |