| 1 |
32341465 | Diabetes downregulates peptide transporter 1 in the rat jejunum: possible involvement of cholate-induced FXR activation. | 2020 Nov |
1 |
| 2 |
29580877 | Establishment of a novel microscale thermophoresis ligand-binding assay for characterization of SLC solute carriers using oligopeptide transporter PepT1 (SLC15 family) as a model system. | 2018 Jul - Aug |
1 |
| 3 |
27719884 | Effect of molecular weight on the transepithelial transport and peptidase degradation of casein-derived peptides by using Caco-2 cell model. | 2017 Mar 1 |
1 |
| 4 |
26924013 | Structural Design of Oligopeptides for Intestinal Transport Model. | 2016 Mar 16 |
1 |
| 5 |
27547863 | The Role of N-Glycosylation in Maintaining the Transporter Activity and Expression of Human Oligopeptide Transporter 1. | 2016 Oct 3 |
2 |
| 6 |
25178856 | Intestinal transport of TRH analogs through PepT1: the role of in silico and in vitro modeling. | 2014 Oct |
3 |
| 7 |
23962042 | Sertraline inhibits the transport of PAT1 substrates in vivo and in vitro. | 2013 Nov |
1 |
| 8 |
22369721 | Construction, identification and application of HeLa cells stably transfected with human PEPT1 and PEPT2. | 2012 Apr |
5 |
| 9 |
22779445 | Mechanistic insights into PEPT1-mediated transport of a novel antiepileptic, NP-647. | 2012 Sep 4 |
1 |
| 10 |
22842481 | The PepT1-transportable soy tripeptide VPY reduces intestinal inflammation. | 2012 Nov |
1 |
| 11 |
21147219 | Affinity and translocation relationships via hPEPT1 of H-X aa-Ser-OH dipeptides: evaluation of H-Phe-Ser-OH as a pro-moiety for ibuprofen and benzoic acid prodrugs. | 2011 Feb |
1 |
| 12 |
21262302 | Uptake, transport and regulation of JBP485 by PEPT1 in vitro and in vivo. | 2011 Apr |
1 |
| 13 |
21280612 | Bifunctional peptidomimetic prodrugs of didanosine for improved intestinal permeability and enhanced acidic stability: synthesis, transepithelial transport, chemical stability and pharmacokinetics. | 2011 Apr 4 |
1 |
| 14 |
21529830 | Differentiating passive from transporter-mediated uptake by PepT1: a comparison and evaluation of four methods. | 2011 Sep |
2 |
| 15 |
21703856 | The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1. | 2011 Aug 1 |
1 |
| 16 |
20128809 | Delta-aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1). | 2010 Mar |
1 |
| 17 |
20307658 | Inhibition of oligopeptide transporter suppress growth of human pancreatic cancer cells. | 2010 Jun 14 |
2 |
| 18 |
20449699 | A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1). | 2010 Sep |
1 |
| 19 |
20558765 | PepT1 mediates transport of the proinflammatory bacterial tripeptide L-Ala-{gamma}-D-Glu-meso-DAP in intestinal epithelial cells. | 2010 Sep |
1 |
| 20 |
20726987 | Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen. | 2010 Dec |
4 |
| 21 |
20929265 | Serine side chain-linked peptidomimetic conjugates of cyclic HPMPC and HPMPA: synthesis and interaction with hPEPT1. | 2010 Dec 6 |
1 |
| 22 |
18781650 | Peptide derivation of poorly absorbable drug allows intestinal absorption via peptide transporter. | 2009 May |
2 |
| 23 |
19115956 | Synthesis, transport and pharmacokinetics of 5'-amino acid ester prodrugs of 1-beta-D-arabinofuranosylcytosine. | 2009 Jan-Feb |
1 |
| 24 |
19201665 | Rapid and sensitive hydrophilic interaction chromatography/tandem mass spectrometry method for the determination of glycyl-sarcosine in cell homogenates. | 2009 Mar 1 |
2 |
| 25 |
19685173 | Mutagenesis and cysteine scanning of transmembrane domain 10 of the human dipeptide transporter. | 2009 Oct |
1 |
| 26 |
27713232 | Effect of Different Metal Ions on the Biological Properties of Cefadroxil. | 2009 Dec 15 |
2 |
| 27 |
18094991 | hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3. | 2008 Jun |
2 |
| 28 |
18336632 | Ethanol inhibits functional activity of the human intestinal dipeptide transporter hPepT1 expressed in Xenopus oocytes. | 2008 May |
1 |
| 29 |
18782614 | Comparison of drug transporter gene expression and functionality in Caco-2 cells from 10 different laboratories. | 2008 Dec 18 |
2 |
| 30 |
17009102 | A charge pair interaction between Arg282 in transmembrane segment 7 and Asp341 in transmembrane segment 8 of hPepT1. | 2007 Jan |
7 |
| 31 |
17407174 | Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1. | 2007 Apr |
2 |
| 32 |
17554807 | Transport of a tripeptide, Gly-Pro-Hyp, across the porcine intestinal brush-border membrane. | 2007 Jul |
1 |
| 33 |
17944948 | Synthesis and characterization of a new and radiolabeled high-affinity substrate for H+/peptide cotransporters. | 2007 Nov |
1 |
| 34 |
16283203 | Prediction of glycylsarcosine transport in Caco-2 cell lines expressing PEPT1 at different levels. | 2006 Apr |
3 |
| 35 |
16328452 | Tumor necrosis factor-alpha and interferon-gamma increase PepT1 expression and activity in the human colon carcinoma cell line Caco-2/bbe and in mouse intestine. | 2006 Apr |
1 |
| 36 |
16568107 | hPepT1 mediates bacterial tripeptide fMLP uptake in human monocytes. | 2006 May |
1 |
| 37 |
16627568 | Molecular interactions between dipeptides, drugs and the human intestinal H+ -oligopeptide cotransporter hPEPT1. | 2006 Jul 1 |
2 |
| 38 |
16651734 | The extracellular pH dependency of transport activity by human oligopeptide transporter 1 (hPEPT1) expressed stably in Chinese hamster ovary (CHO) cells: a reason for the bell-shaped activity versus pH. | 2006 May |
2 |
| 39 |
16713701 | In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1. | 2006 Jul |
2 |
| 40 |
15623827 | Alanylglutamine dipeptide and growth hormone maintain PepT1-mediated transport in oxidatively stressed Caco-2 cells. | 2005 Jan |
1 |
| 41 |
15340850 | Efflux properties of basolateral peptide transporter in human intestinal cell line Caco-2. | 2004 Nov |
1 |
| 42 |
15521010 | hPepT1 transports muramyl dipeptide, activating NF-kappaB and stimulating IL-8 secretion in human colonic Caco2/bbe cells. | 2004 Nov |
1 |
| 43 |
15832510 | A novel hPepT1 stably transfected cell line: establishing a correlation between expression and function. | 2004 Mar-Apr |
2 |
| 44 |
15981923 | Comparison of human and monkey peptide transporters: PEPT1 and PEPT2. | 2004 May-Jun |
2 |
| 45 |
12788085 | Transmembrane segment 5 of the dipeptide transporter hPepT1 forms a part of the substrate translocation pathway. | 2003 Jun 20 |
1 |
| 46 |
14532279 | Analysis of transmembrane segment 7 of the dipeptide transporter hPepT1 by cysteine-scanning mutagenesis. | 2003 Dec 19 |
2 |
| 47 |
14661916 | A fluorescent hPept1 transporter substrate for uptake screening. | 2003 Nov |
2 |
| 48 |
14725353 | Biophysical evidence for His57 as a proton-binding site in the mammalian intestinal transporter hPepT1. | 2003 Dec |
4 |
| 49 |
12009949 | Inhibitory effect of supramolecular polyrotaxane-dipeptide conjugates on digested peptide uptake via intestinal human peptide transporter. | 2002 May-Jun |
1 |
| 50 |
11459451 | Significance of substrate hydrophobicity for recognition by an oligopeptide transporter (PEPT1). | 2001 Jul-Aug |
1 |