Title : Bifunctional peptidomimetic prodrugs of didanosine for improved intestinal permeability and enhanced acidic stability: synthesis, transepithelial transport, chemical stability and pharmacokinetics.

Pub. Date : 2011 Apr 4

PMID : 21280612

1 Functional Relationships(s)
Compound Name
Protein Name
1 The uptake of glycylsarcosine (Gly-Sar, a typical substrate of PepT1) by Caco-2 cells could be inhibited by compound 4a in a concentration-dependent manner. Glycine solute carrier family 15 member 1 Homo sapiens