Salmeterol Xinafoate

adrenoceptor beta 2 ; Homo sapiens







122 Article(s)
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1 34334369 Membrane-Facilitated Receptor Access and Binding Mechanisms of Long-Acting β2-Adrenergic Receptor Agonists. 2021 Oct 1
2 29653961 Analysis of the Indacaterol-Regulated Transcriptome in Human Airway Epithelial Cells Implicates Gene Expression Changes in the Adverse and Therapeutic Effects of β2-Adrenoceptor Agonists. 2018 Jul 2
3 30327561 Structural insights into binding specificity, efficacy and bias of a β2AR partial agonist. 2018 Nov 4
4 28097668 Detection and pharmacokinetics of salmeterol in thoroughbred horses following inhaled administration. 2017 Oct 1
5 28398147 Salmeterol, a Long-Acting β2-Adrenergic Receptor Agonist, Inhibits Macrophage Activation by Lipopolysaccharide From Porphyromonas gingivalis. 2017 Jul 2
6 27222010 Sympathetic neural signaling via the β2-adrenergic receptor suppresses T-cell receptor-mediated human and mouse CD8(+) T-cell effector function. 2016 Aug 1
7 27885204 GENETIC INTERACTIONS BETWEEN ADRB2 AND PTGER4 ON RESPONSES TO SALMETEROL OR MONTELUKAST IN JAPANESE PATIENTS WITH MILD PERSISTENT ASTHMA. 2016 2
8 25324048 Salmeterol's extreme β2 selectivity is due to residues in both extracellular loops and transmembrane domains. 2015 Jan 1
9 25784721 Salmeterol Efficacy and Bias in the Activation and Kinase-Mediated Desensitization of β2-Adrenergic Receptors. 2015 Jun 5
10 25799096 ASM-024, a piperazinium compound, promotes the in vitro relaxation of β2-adrenoreceptor desensitized tracheas. 2015 1
11 26049917 Why use long acting bronchodilators in chronic obstructive lung diseases? An extensive review on formoterol and salmeterol. 2015 Jul 1
12 26051688 Salmeterol Xinafoate. 2015 1
13 24461901 Effect of ADRB2 polymorphisms on the efficacy of salmeterol and tiotropium in preventing COPD exacerbations: a prespecified substudy of the POET-COPD trial. 2014 Jan 1
14 24561123 CHIP-MYTH: a novel interactive proteomics method for the assessment of agonist-dependent interactions of the human β₂-adrenergic receptor. 2014 Mar 21 1
15 24681963 The effects of a Gly16Arg ADRB2 polymorphism on responses to salmeterol or montelukast in Japanese patients with mild persistent asthma. 2014 May 1
16 24721141 Effect of β2 -adrenergic receptor gene Arg16Gly polymorphisms on response to long-acting β2-agonist in Chinese Han asthmatic patients. 2014 1
17 23302644 Agonist-induced receptor internalization in Chinese hamster ovary cells stably co-expressing β(1)- and β(2)-adrenergic receptors. 2013 6
18 23375225 Hybrids consisting of the pharmacophores of salmeterol and roflumilast or phthalazinone: dual β₂-adrenoceptor agonists-PDE4 inhibitors for the treatment of COPD. 2013 Mar 1 2
19 23548523 Influence of β(2)-adrenergic receptor polymorphisms on asthma exacerbation in children with severe asthma regularly receiving salmeterol. 2013 Mar 1
20 24228710 Loss of salmeterol bronchoprotection against exercise in relation to ADRB2 Arg16Gly polymorphism and exhaled nitric oxide. 2013 Dec 15 1
21 22306235 Additive anti-inflammatory effects of beta 2 adrenoceptor agonists or glucocorticosteroid with roflumilast in human peripheral blood mononuclear cells. 2012 Apr 1
22 23131487 Lactic acidosis following intentional overdose by inhalation of salmeterol and fluticasone. 2012 Nov 1
23 23300522 Identifying ligand binding conformations of the β2-adrenergic receptor by using its agonists as computational probes. 2012 2
24 21134482 The reassertion profiles of long acting β2-adrenoceptor agonists in the guinea pig isolated trachea and human recombinant β2-adrenoceptor. 2011 Apr 2
25 21306583 Formoterol and salmeterol induce a similar degree of β2-adrenoceptor tolerance in human small airways but via different mechanisms. 2011 Jun 1
26 21357659 Functional and biochemical rationales for the 24-hour-long duration of action of olodaterol. 2011 Jun 1
27 20003162 Suppressive effects of formoterol and salmeterol on eotaxin-1 in bronchial epithelial cells. 2010 Mar 1
28 20423350 Enhancement of inflammatory mediator release by beta(2)-adrenoceptor agonists in airway epithelial cells is reversed by glucocorticoid action. 2010 May 1
29 20590599 The selectivity of beta-adrenoceptor agonists at human beta1-, beta2- and beta3-adrenoceptors. 2010 Jul 1
30 19059194 Beta2-adrenoreceptor ligands regulate osteoclast differentiation in vitro by direct and indirect mechanisms. 2009 Feb 1
31 19201814 Modulation of epidermal growth factor receptor binding to human airway smooth muscle cells by glucocorticoids and beta2-adrenergic receptor agonists. 2009 Apr 1
32 19594756 Molecular mechanisms for the persistent bronchodilatory effect of the beta 2-adrenoceptor agonist salmeterol. 2009 Sep 1
33 19666775 Mechanism regulating proasthmatic effects of prolonged homologous beta2-adrenergic receptor desensitization in airway smooth muscle. 2009 Oct 2
34 19719334 Salmeterol/fluticasone propionate: a review of its use in asthma. 2009 1
35 19719779 Agonist efficacy and receptor desensitization: from partial truths to a fuller picture. 2009 Sep 1
36 19800676 Adrenergic beta(2)-receptor genotype predisposes to exacerbations in steroid-treated asthmatic patients taking frequent albuterol or salmeterol. 2009 Dec 2
37 17901197 Long-acting beta2-adrenoceptor agonists synergistically enhance glucocorticoid-dependent transcription in human airway epithelial and smooth muscle cells. 2008 Jan 1
38 17993585 Inhibition of human airway smooth muscle cell proliferation by beta 2-adrenergic receptors and cAMP is PKA independent: evidence for EPAC involvement. 2008 Jan 1
39 18512086 An insilico approach to high altitude pulmonary edema - Molecular modeling of human beta2 adrenergic receptor and its interaction with Salmeterol & Nifedipine. 2008 Sep 3
40 18586957 Effect of beta2-adrenoceptor agonists and other cAMP-elevating agents on inflammatory gene expression in human ASM cells: a role for protein kinase A. 2008 Sep 1
41 16980556 Salmeterol stimulation dissociates beta2-adrenergic receptor phosphorylation and internalization. 2007 Feb 4
42 17631879 Combination of fluticasone propionate and salmeterol potentiates the suppression of cigarette smoke-induced IL-8 production by macrophages. 2007 Sep 24 1
43 17846318 A novel role of the sympatho-adrenergic system in regulating valve calcification. 2007 Sep 11 1
44 16772309 Arginine-16 beta2 adrenoceptor genotype predisposes to exacerbations in young asthmatics taking regular salmeterol. 2006 Nov 1
45 17030231 Salmeterol response is not affected by beta2-adrenergic receptor genotype in subjects with persistent asthma. 2006 Oct 2
46 15655528 The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors. 2005 Feb 1
47 16022567 Ultra long-acting beta 2-agonists in development for asthma and chronic obstructive pulmonary disease. 2005 Jul 1
48 14662724 Desensitisation of mast cell beta2-adrenoceptor-mediated responses by salmeterol and formoterol. 2004 Jan 5
49 14678342 The arginine-16 beta2-adrenoceptor polymorphism predisposes to bronchoprotective subsensitivity in patients treated with formoterol and salmeterol. 2004 Jan 1
50 15182210 Redefining treatment in COPD: new directions in bronchodilator therapy. 2004 1