Amides

ETS transcription factor ERG ; Homo sapiens







10 Article(s)
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Pub. Year
#Total Relationships
1 34413963 Structure-Activity Relationship Studies Reveal New Astemizole Analogues Active against Plasmodium falciparum In Vitro. 2021 Aug 12 1
2 26804230 Optimization of tetrahydronaphthalene inhibitors of Raf with selectivity over hERG. 2016 Feb 15 1
3 26141771 Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6). 2015 Sep 1 1
4 24412109 Successful reduction of off-target hERG toxicity by structural modification of a T-type calcium channel blocker. 2014 Feb 1 1
5 24486132 IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: improved PK, hERG and metabolic profiles. 2014 Feb 15 1
6 21414780 Novel pyrrolidine melanin-concentrating hormone receptor 1 antagonists with reduced hERG inhibition. 2011 Apr 15 1
7 21515049 Macrocyclic lactams as potent Hsp90 inhibitors with excellent tumor exposure and extended biomarker activity. 2011 Jun 1 1
8 20570511 Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors. 2010 Jul 15 1
9 20684603 Discovery of 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidine-2-carboxamides as potent, selective dipeptidyl peptidase-4 (DPP4) inhibitors. 2010 Aug 12 1
10 19821563 Structure-activity relationships of 9-substituted-9-dihydroerythromycin-based motilin agonists: optimizing for potency and safety. 2009 Nov 12 1