Fenoterol

adrenoceptor beta 2 ; Homo sapiens







56 Article(s)
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1 28338133 Stereoselective binding of agonists to the β2-adrenergic receptor: insights into molecular details and thermodynamics from molecular dynamics simulations. 2017 May 2 3
2 28603032 β2-adrenergic receptor-mediated in vitro regulation of human hepatic drug transporter expression by epinephrine. 2017 Aug 30 1
3 27657826 Anti-inflammatory activities of fenoterol through β-arrestin-2 and inhibition of AMPK and NF-κB activation in AICAR-induced THP-1 cells. 2016 Dec 2
4 25342094 Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the β2-adrenoceptor. 2015 Jan 2
5 25637582 Interaction of fenoterol stereoisomers with β2-adrenoceptor-G sα fusion proteins: antagonist and agonist competition binding. 2015 May 4
6 25930996 Fenoterol inhibits LPS-induced AMPK activation and inflammatory cytokine production through β-arrestin-2 in THP-1 cell line. 2015 Jun 26 3
7 24182991 The β2-adrenoreceptor gene promoter polymorphisms may modulate β2-agonist- and glucocorticoid-induced IgE synthesis. 2014 Nov-Dec 2
8 24326276 Comparative molecular field analysis of fenoterol derivatives interacting with an agonist-stabilized form of the β₂-adrenergic receptor. 2014 Jan 1 3
9 24441217 Stereochemical and conformational study on fenoterol by ECD spectroscopy and TD-DFT calculations. 2014 Mar 4
10 24615679 Fast, metadynamics-based method for prediction of the stereochemistry-dependent relative free energies of ligand-receptor interactions. 2014 Apr 30 2
11 24633512 Oriented immobilisation of histidine-tagged protein and its application in exploring interactions between ligands and proteins. 2014 May 2
12 25360795 Wnt/β-catenin signaling modulates human airway sensitization induced by β2-adrenoceptor stimulation. 2014 1
13 24043542 Molecular interactions between fenoterol stereoisomers and derivatives and the β₂-adrenergic receptor binding site studied by docking and molecular dynamics simulations. 2013 Nov 4
14 22434858 Thermodynamics and docking of agonists to the β(2)-adrenoceptor determined using [(3)H](R,R')-4-methoxyfenoterol as the marker ligand. 2012 Jun 2
15 22760074 Fenoterol functionally activates the β₃-adrenoceptor in human urinary bladder, comparison with rat and mouse: implications for drug discovery. 2012 Sep 5 2
16 22776956 Cannabinoid receptor activation correlates with the proapoptotic action of the β2-adrenergic agonist (R,R')-4-methoxy-1-naphthylfenoterol in HepG2 hepatocarcinoma cells. 2012 Oct 4
17 21320165 Inhibitory effects of albuterol and fenoterol on RANTES and IP-10 expression in bronchial epithelial cells. 2011 Jun 1
18 21365223 Modeling of ligand binding to G protein coupled receptors: cannabinoid CB1, CB2 and adrenergic β 2 AR. 2011 Sep 1
19 20036561 Comparative molecular field analysis of fenoterol derivatives: A platform towards highly selective and effective beta(2)-adrenergic receptor agonists. 2010 Jan 15 1
20 20144591 The effect of stereochemistry on the thermodynamic characteristics of the binding of fenoterol stereoisomers to the beta(2)-adrenoceptor. 2010 Jun 1 4
21 20837485 Differential signaling of the endogenous agonists at the beta2-adrenergic receptor. 2010 Nov 12 2
22 18838481 Stereochemistry of an agonist determines coupling preference of beta2-adrenoceptor to different G proteins in cardiomyocytes. 2009 Jan 1
23 19462961 Peroxidative metabolism of beta2-agonists salbutamol and fenoterol and their analogues. 2009 Jun 1
24 19703961 Laminin enhances beta(2)-adrenergic receptor stimulation of L-type Ca(2+) current via cytosolic phospholipase A(2) signalling in cat atrial myocytes. 2009 Oct 15 2
25 19890360 Fenoterol, a beta(2)-adrenoceptor agonist, inhibits LPS-induced membrane-bound CD14, TLR4/CD14 complex, and inflammatory cytokines production through beta-arrestin-2 in THP-1 cell line. 2009 Nov 2
26 18641310 Low- versus high-baseline epinephrine output shapes opposite innate cytokine profiles: presence of Lewis- and Fischer-like neurohormonal immune phenotypes in humans? 2008 Aug 1 1
27 17506540 Comparative molecular field analysis of the binding of the stereoisomers of fenoterol and fenoterol derivatives to the beta2 adrenergic receptor. 2007 Jun 14 3
28 16448568 Limited beta2-adrenoceptor haplotypes display different agonist mediated airway responses in asthmatics. 2006 Jan 31 1
29 16917835 Enantioselective separation and online affinity chromatographic characterization of R,R- and S,S-fenoterol. 2006 Nov 4
30 15715182 Past, present and future--beta2-adrenoceptor agonists in asthma management. 2005 Feb 1
31 15728216 Self-limitation of intravenous tocolysis with beta2-adrenergic agonists is mediated through receptor G protein uncoupling. 2005 May 1
32 15965358 Ligands at beta2-, beta3-, and the low-affinity state of beta1-adrenoceptors block the alpha1-adrenoceptor-mediated constriction in human pulmonary and rat mesenteric arteries. 2005 Jul 1
33 16147906 Beta2-adrenoceptor agonists induce the mammalian clock gene, hPer1, mRNA in cultured human bronchial epithelium cells in vitro. 2005 1
34 15351928 Nociceptin inhibits vanilloid TRPV-1-mediated neurosensitization induced by fenoterol in human isolated bronchi. 2004 Sep 1
35 12154173 Nitric oxide signalling by selective beta(2)-adrenoceptor stimulation prevents ACh-induced inhibition of beta(2)-stimulated Ca(2+) current in cat atrial myocytes. 2002 Aug 1 2
36 12452831 Inhibition by fenoterol of human eosinophil functions including beta2-adrenoceptor-independent actions. 2002 Dec 1
37 11755157 RANTES release by human airway smooth muscle: effects of prostaglandin E(2) and fenoterol. 2001 Dec 21 1
38 10464825 beta 2-agonist-induced inhibition of neutrophil chemotaxis is not associated with modification of LFA-1 and Mac-1 expression or with impairment of polymorphonuclear leukocyte antibacterial activity. 1999 Jun 1
39 9730867 Beta-adrenoceptor-mediated inhibition of IFN-gamma, IL-3, and GM-CSF mRNA accumulation in activated human T lymphocytes is solely mediated by the beta2-adrenoceptor subtype. 1998 Sep 1
40 9734347 Downregulation of the expression of intercellular adhesion molecule (ICAM)-1 on bronchial epithelial cells by fenoterol, a beta2-adrenoceptor agonist. 1998 1
41 9056046 Evaluation of partial beta-adrenoceptor agonist activity. 1997 Jan 1
42 9209250 Fenoterol but not dobutamine increases erythropoietin production in humans. 1997 Jun 1
43 9295336 beta2-adrenergic receptor desensitization, internalization, and phosphorylation in response to full and partial agonists. 1997 Sep 19 3
44 8730730 Anti-inflammatory, membrane-stabilizing interactions of salmeterol with human neutrophils in vitro. 1996 Apr 1
45 8777955 Role of cyclic AMP in the modulation of IgE production by the beta 2-adrenoceptor agonist, fenoterol. 1996 Feb 1
46 8911881 Concentration-effect relationship of the positive chronotropic and hypokalaemic effects of fenoterol in healthy women of childbearing age. 1996 1
47 8094228 Functional interaction between beta 2-adrenoceptor agonists and interleukin-4 in the regulation of CD23 expression and release and IgE production in human. 1993 Feb 1
48 8103795 Thermoregulatory effects of beta adrenoceptors: effects of selective agonists and the interaction of antagonists with isoproterenol and BRL-35135 in the cold. 1993 Sep 1
49 1348446 Reduced alpha 1- and beta 2-adrenoceptor-mediated positive inotropic effects in human end-stage heart failure. 1992 Feb 1
50 1493852 The pharmacokinetics of the beta 2-adrenoceptor agonist fenoterol in healthy women. 1992 1