Title : Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the β2-adrenoceptor.

Pub. Date : 2015 Jan

PMID : 25342094






2 Functional Relationships(s)
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1 Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the beta2-adrenoceptor. Fenoterol adrenoceptor beta 2 Homo sapiens
2 Ligand bias was calculated using an operational model of agonism and revealed that the fenoterol scaffold constitutes a promising lead structure for the development of Gs-biased beta2AR agonists. Fenoterol adrenoceptor beta 2 Homo sapiens