enzalutamide

androgen receptor ; Homo sapiens







487 Article(s)
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1 34449248 A New Old Target: Androgen Receptor Signaling and Advanced Prostate Cancer. 2022 Jan 6 3
2 34648657 A European, prospective, observational study of enzalutamide in patients with metastatic castration-resistant prostate cancer: PREMISE. 2022 Mar 1 1
3 34728570 Targeting DNMTs to Overcome Enzalutamide Resistance in Prostate Cancer. 2022 Jan 2
4 34740892 Loss of Long Noncoding RNA NXTAR in Prostate Cancer Augments Androgen Receptor Expression and Enzalutamide Resistance. 2022 Jan 1 3
5 34763937 Phase II study of enzalutamide in androgen receptor positive, recurrent, high- and low-grade serous ovarian cancer. 2022 Jan 2
6 34807458 Phase I clinical trial of HC-1119 soft capsule in Chinese healthy adult male subjects: Pharmacokinetics and safety of single-dose proportionality and effects of food. 2022 Feb 3
7 34937944 Targeting SWI/SNF ATPases in enhancer-addicted prostate cancer. 2022 Jan 1
8 35058329 (+)-JJ-74-138 is a Novel Noncompetitive Androgen Receptor Antagonist. 2022 Apr 1 3
9 35229000 Prognostic significance of risk stratification in CHAARTED and LATITUDE studies among Japanese men with castration-resistant prostate cancer. 2022 Mar 1
10 35271265 Application of Surface-Enhanced Raman Spectroscopy to Guide Therapy for Advanced Prostate Cancer Patients. 2022 Mar 25 3
11 35337811 Chemical degrader enhances the treatment of androgen receptor-positive triple-negative breast cancer. 2022 May 30 1
12 35352309 Real-World Effectiveness of Sipuleucel-T on Overall Survival in Men with Advanced Prostate Cancer Treated with Androgen Receptor-Targeting Agents. 2022 Jun 1
13 35363301 Phase Ib/II Study of Enzalutamide with Samotolisib (LY3023414) or Placebo in Patients with Metastatic Castration-Resistant Prostate Cancer. 2022 Jun 1 1
14 35372002 Prognostic and Predictive Value of Liquid Biopsy-Derived Androgen Receptor Variant 7 (AR-V7) in Prostate Cancer: A Systematic Review and Meta-Analysis. 2022 1
15 35372068 Anti-Androgen Receptor Therapies in Prostate Cancer: A Brief Update and Perspective. 2022 1
16 35385726 Mesenchymal and stem-like prostate cancer linked to therapy-induced lineage plasticity and metastasis. 2022 Apr 5 2
17 35390118 Targeting the androgen receptor signaling pathway in advanced prostate cancer. 2022 Apr 7 2
18 35428760 RNF8 up-regulates AR/ARV7 action to contribute to advanced prostate cancer progression. 2022 Apr 15 1
19 35452181 Both SUMOylation and ubiquitination of TFE3 fusion protein regulated by androgen receptor are the potential target in the therapy of Xp11.2 translocation renal cell carcinoma. 2022 Apr 2
20 35504877 Non-drug efflux function of ABCC5 promotes enzalutamide resistance in castration-resistant prostate cancer via upregulation of P65/AR-V7. 2022 May 3 1
21 35510101 Prognostic impact of dose reduction in androgen receptor pathway inhibitors for castration-resistant prostate cancer. 2022 Mar 1
22 35513478 Grade group system and plasma androgen receptor status in the first line treatment for metastatic castration resistant prostate cancer. 2022 May 5 4
23 35523048 Antagonistic action of a synthetic androgen ligand mediated by chromatin remodeling in a human prostate cancer cell line. 2022 Jul 5 6
24 35533600 Lycopene enhances the sensitivity of castration-resistant prostate cancer to enzalutamide through the AKT/EZH2/ androgen receptor signaling pathway. 2022 Jul 12 2
25 35534851 Natural product myricetin is a pan-KDM4 inhibitor which with poly lactic-co-glycolic acid formulation effectively targets castration-resistant prostate cancer. 2022 May 9 1
26 35553247 Decisions and dilemmas in non-metastatic castration-resistant prostate cancer management. 2022 May 13 1
27 35565349 Baseline Plasma Tumor DNA (ctDNA) Correlates with PSA Kinetics in Metastatic Castration-Resistant Prostate Cancer (mCRPC) Treated with Abiraterone or Enzalutamide. 2022 Apr 29 1
28 35579577 Factors that guide selection among androgen receptor inhibitors in patients with nonmetastatic castration-resistant prostate cancer. 2022 May 1
29 35590370 The DNA/RNA helicase DHX9 contributes to the transcriptional program of the androgen receptor in prostate cancer. 2022 May 19 1
30 31558422 Progression-directed Therapy for Oligoprogression in Castration-refractory Prostate Cancer. 2021 Apr 1
31 31676281 Improved Androgen Receptor Splice Variant 7 Detection Using a Highly Sensitive Assay to Predict Resistance to Abiraterone or Enzalutamide in Metastatic Prostate Cancer Patients. 2021 Aug 2
32 32624280 A Multicohort Open-label Phase II Trial of Bipolar Androgen Therapy in Men with Metastatic Castration-resistant Prostate Cancer (RESTORE): A Comparison of Post-abiraterone Versus Post-enzalutamide Cohorts. 2021 May 1
33 32881669 Darolutamide as a Second-Generation Androgen Receptor Inhibitor in the Treatment of Prostate Cancer. 2021 1
34 32954481 Isolation and characterization of castration-resistant prostate cancer LNCaP95 clones. 2021 Jan 3
35 32958445 Androgen receptor inhibitor treatments: Cardiovascular adverse events and comorbidity considerations in patients with non-metastatic prostate cancer. 2021 Jan 1
36 33140306 Endocrine consequences of treatment with the new androgen receptor axis-targeted agents for advanced prostate cancer. 2021 Mar 1
37 33150960 Mechanisms of enzalutamide resistance in castration-resistant prostate cancer and therapeutic strategies to overcome it. 2021 Jan 3
38 33271252 Functional characterization of androgen receptor in two patient-derived xenograft models of triple negative breast cancer. 2021 Feb 1
39 33277366 KIF15-Mediated Stabilization of AR and AR-V7 Contributes to Enzalutamide Resistance in Prostate Cancer. 2021 Feb 15 4
40 33277796 A review of the effects and molecular mechanisms of dimethylcurcumin (ASC-J9) on androgen receptor-related diseases. 2021 Apr 1
41 33388655 Design, synthesis and biological evaluation of novel thiohydantoin derivatives as potent androgen receptor antagonists for the treatment of prostate cancer. 2021 Feb 1 3
42 33432555 Clinicopathological Features and Treatment Challenges in Triple Negative Breast Cancer Patients: A Retrospective Cohort Study. 2021 2
43 33436326 Circulating Androgen Receptor for Prognosis and Treatment Selection in Prostate Cancer. 2021 Oct 3
44 33441906 Regulation of carcinogenesis and mediation through Wnt/β-catenin signaling by 3,3'-diindolylmethane in an enzalutamide-resistant prostate cancer cell line. 2021 Jan 13 4
45 33470111 Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC). 2021 Jan 28 2
46 33500577 Androgen receptor gain in circulating free DNA and splicing variant 7 in exosomes predict clinical outcome in CRPC patients treated with abiraterone and enzalutamide. 2021 Jun 1
47 33517325 Synthesis and Evaluation of 18F-Enzalutamide, a New Radioligand for PET Imaging of Androgen Receptors: A Comparison with 16β-18F-Fluoro-5α-Dihydrotestosterone. 2021 Aug 1 3
48 33562646 Metformin and Androgen Receptor-Axis-Targeted (ARAT) Agents Induce Two PARP-1-Dependent Cell Death Pathways in Androgen-Sensitive Human Prostate Cancer Cells. 2021 Feb 5 1
49 33563753 V-ATPase Inhibition Decreases Mutant Androgen Receptor Activity in Castrate-resistant Prostate Cancer. 2021 Apr 3
50 33574348 Inhibition of androgen/AR signaling inhibits diethylnitrosamine (DEN) induced tumour initiation and remodels liver immune cell networks. 2021 Feb 11 1