5 Article(s)Download |
PMID | Title | Pub. Year | #Total Relationships |
1 | 21220496 | Drug efflux by breast cancer resistance protein is a mechanism of resistance to the benzimidazole insulin-like growth factor receptor/insulin receptor inhibitor, BMS-536924. | 2011 Jan | 1 |
2 | 20153189 | SAR of PXR transactivation in benzimidazole-based IGF-1R kinase inhibitors. | 2010 Mar 1 | 1 |
3 | 20545947 | Design of potent IGF1-R inhibitors related to bis-azaindoles. | 2010 Aug | 1 |
4 | 18572407 | Balancing oral exposure with Cyp3A4 inhibition in benzimidazole-based IGF-IR inhibitors. | 2008 Jul 15 | 1 |
5 | 18763755 | Discovery and evaluation of 4-(2-(4-chloro-1H-pyrazol-1-yl)ethylamino)-3-(6-(1-(3-fluoropropyl)piperidin-4-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one (BMS-695735), an orally efficacious inhibitor of insulin-like growth factor-1 receptor kinase with broad spectrum in vivo antitumor activity. | 2008 Oct 9 | 1 |