| 1 |
34021071 | Defining the Energetic Basis for a Conformational Switch Mediating Ligand-Independent Activation of Mutant Estrogen Receptors in Breast Cancer. | 2021 Sep |
2 |
| 2 |
34073781 | β-Sitosterol-D-Glucopyranoside Mimics Estrogenic Properties and Stimulates Glucose Utilization in Skeletal Muscle Cells. | 2021 May 24 |
1 |
| 3 |
31602686 | Investigation of binding mechanism and downregulation of elacestrant for wild and L536S mutant estrogen receptor-α through molecular dynamics simulation and binding free energy analysis. | 2020 Jan 15 |
1 |
| 4 |
32344252 | Assessment of endocrine-disrupting effects of emerging polyhalogenated carbazoles (PHCZs): In vitro, in silico, and in vivo evidence. | 2020 Jul |
2 |
| 5 |
32705198 | Antitumor effects of aconitine in A2780 cells via estrogen receptor β‑mediated apoptosis, DNA damage and migration. | 2020 Sep |
1 |
| 6 |
29557271 | Structural insight into the antagonistic action of diarylheptanoid on human estrogen receptor alpha. | 2019 Mar |
1 |
| 7 |
30587451 | Selective estrogen receptor degraders with novel structural motifs induce regression in a tamoxifen-resistant breast cancer xenograft. | 2019 Feb 1 |
1 |
| 8 |
29392883 | In silico binding of 4,4'-bisphenols predicts in vitro estrogenic and antiandrogenic activity. | 2018 May |
2 |
| 9 |
29587221 | Structure-activity relationships of 2, 4-disubstituted pyrimidines as dual ERα/VEGFR-2 ligands with anti-breast cancer activity. | 2018 Apr 25 |
1 |
| 10 |
28216037 | ESR1 single nucleotide polymorphism rs1062577 (c.*3804T>A) alters the susceptibility of breast cancer risk in Iranian population. | 2017 May 5 |
1 |
| 11 |
27589781 | Phytoestrogens and Mycoestrogens Induce Signature Structure Dynamics Changes on Estrogen Receptor α. | 2016 Aug 31 |
1 |
| 12 |
27743518 | Estrogen Receptor Binding Affinity of Food Contact Material Components Estimated by QSAR. | 2016 Sep |
1 |
| 13 |
26308263 | Estrogenic activity data extraction and in silico prediction show the endocrine disruption potential of bisphenol A replacement compounds. | 2015 Sep 21 |
1 |
| 14 |
24315190 | Probing the human estrogen receptor-α binding requirements for phenolic mono- and di-hydroxyl compounds: a combined synthesis, binding and docking study. | 2014 Jan 1 |
1 |
| 15 |
24507131 | Molecular docking and molecular dynamics studies on the interactions of hydroxylated polybrominated diphenyl ethers to estrogen receptor alpha. | 2014 Mar |
1 |
| 16 |
24725156 | Charge clamps of lysines and hydrogen bonds play key roles in the mechanism to fix helix 12 in the agonist and antagonist positions of estrogen receptor α: intramolecular interactions studied by the ab initio fragment molecular orbital method. | 2014 May 15 |
1 |
| 17 |
23200735 | Effects of quercetin on mRNA expression of steroidogenesis genes in primary cultures of Leydig cells treated with atrazine. | 2013 Mar |
1 |
| 18 |
23273518 | Novel Aza-resveratrol analogs: synthesis, characterization and anticancer activity against breast cancer cell lines. | 2013 Feb 1 |
1 |
| 19 |
22503158 | Docking and QSAR study on the binding interactions between polycyclic aromatic hydrocarbons and estrogen receptor. | 2012 Jun |
1 |
| 20 |
22582136 | Hydrophobic Interactions Improve Selectivity to ERα for Ben-zothiophene SERMs. | 2012 Mar 8 |
1 |
| 21 |
21163906 | Estrogen-like activity of perfluoroalkyl acids in vivo and interaction with human and rainbow trout estrogen receptors in vitro. | 2011 Mar |
1 |
| 22 |
22061644 | Investigation of the diastereomerism of dihydrobenzoxathiin SERMs for ER alpha by molecular modeling. | 2011 Dec 15 |
1 |
| 23 |
20669983 | Effects of 7-O substitutions on estrogenic and anti-estrogenic activities of daidzein analogues in MCF-7 breast cancer cells. | 2010 Aug 26 |
2 |
| 24 |
19128016 | Structural evolutions of salicylaldoximes as selective agonists for estrogen receptor beta. | 2009 Feb 12 |
3 |
| 25 |
19739677 | Unique ligand binding patterns between estrogen receptor alpha and beta revealed by hydrogen-deuterium exchange. | 2009 Oct 13 |
1 |
| 26 |
18474858 | Prediction of the tissue-specificity of selective estrogen receptor modulators by using a single biochemical method. | 2008 May 20 |
2 |
| 27 |
18591792 | Molecular design based on receptor-independent pharmacophore: application to estrogen receptor ligands. | 2008 Jul |
1 |
| 28 |
17328537 | Pharmacophore mapping of selective binding affinity of estrogen modulators through classical and space modeling approaches: exploration of bridged-cyclic compounds with diarylethylene linkage. | 2007 Mar-Apr |
1 |
| 29 |
16191480 | Targeted mutation of key residues at the start of helix 12 in the hERalpha ligand-binding domain identifies the role of hydrogen-bonding and hydrophobic interactions in the activity of the protein. | 2006 Jan |
1 |
| 30 |
16884312 | Synthesis of anthranylaldoxime derivatives as estrogen receptor ligands and computational prediction of binding modes. | 2006 Aug 10 |
2 |
| 31 |
16898767 | Molecular interactions between estrogen receptor and its ligand studied by the ab initio fragment molecular orbital method. | 2006 Aug 17 |
1 |
| 32 |
15635182 | QSAR studies with E-state index: predicting pharmacophore signals for estrogen receptor binding affinity of triphenylacrylonitriles. | 2005 Jan |
1 |
| 33 |
16326832 | Role of aspartate 351 in transactivation and active conformation of estrogen receptor alpha. | 2005 Dec |
1 |
| 34 |
11708930 | Salicylaldoxime moiety as a phenolic "A-Ring" substitute in estrogen receptor ligands. | 2001 Nov 22 |
2 |
| 35 |
9422719 | Determinants of ligand specificity of estrogen receptor-alpha: estrogen versus androgen discrimination. | 1998 Jan 9 |
2 |
| 36 |
9449681 | The estrogenicity of bisphenol A-related diphenylalkanes with various substituents at the central carbon and the hydroxy groups. | 1998 Mar |
1 |
| 37 |
6292423 | Nonsteroidal estrogens: synthesis and estrogen receptor binding affinity of derivatives of (3R*,4S*)-3,4-bis(4-hydroxyphenyl)hexane (hexestrol) and (2R*,3S*)-2,3-bis(4-hydroxyphenyl)pentane (norhexestrol) functionalized on the side chain. | 1982 Nov |
1 |