Aspartic Acid

estrogen receptor 1 ; Homo sapiens







17 Article(s)
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Title
Pub. Year
#Total Relationships
1 32807064 Synthesis and Evaluation of Cytotoxicity of Novel Coumarin Peptide Alcohol Derivatives. 2021 1
2 29045135 Structural Basis of Inhibition of ERĪ±-Coactivator Interaction by High-Affinity N-Terminus Isoaspartic Acid Tethered Helical Peptides. 2017 Nov 9 1
3 26848530 Human plasma metabolomics for identifying differential metabolites and predicting molecular subtypes of breast cancer. 2016 Mar 1 1
4 16179380 Altered target gene regulation controlled by estrogen receptor-alpha concentration. 2006 Feb 2
5 16191480 Targeted mutation of key residues at the start of helix 12 in the hERalpha ligand-binding domain identifies the role of hydrogen-bonding and hydrophobic interactions in the activity of the protein. 2006 Jan 2
6 16679488 Tamoxifen and raloxifene differ in their functional interactions with aspartate 351 of estrogen receptor alpha. 2006 Aug 1
7 15965534 Identification of the estrogen receptor Cd-binding sites by chemical modification. 2005 Jul 1
8 16326832 Role of aspartate 351 in transactivation and active conformation of estrogen receptor alpha. 2005 Dec 7
9 15604293 Phosphorylation of estrogen receptor alpha blocks its acetylation and regulates estrogen sensitivity. 2004 Dec 15 1
10 12496244 Modulation of estrogen receptor alpha function and stability by tamoxifen and a critical amino acid (Asp-538) in helix 12. 2003 Feb 28 1
11 12790809 Transcriptional activation by estrogen receptor (ERalpha) and steroid receptor coactivator (SRC1) involves distinct mechanisms in yeast and mammalian cells. 2003 Jun 2
12 11751902 Structure-function relationships of the raloxifene-estrogen receptor-alpha complex for regulating transforming growth factor-alpha expression in breast cancer cells. 2002 Mar 15 4
13 11159857 Molecular mechanism of action at estrogen receptor alpha of a new clinically relevant antiestrogen (GW7604) related to tamoxifen. 2001 Feb 2
14 10787412 Aspartate 351 of estrogen receptor alpha is not crucial for the antagonist activity of antiestrogens. 2000 Jul 7 3
15 9581827 The key to the antiestrogenic mechanism of raloxifene is amino acid 351 (aspartate) in the estrogen receptor. 1998 May 1 1
16 9219916 Estrogenic activity is increased for an antiestrogen by a natural mutation of the estrogen receptor. 1997 Mar 1
17 7476979 A naturally occurring estrogen receptor mutation results in increased estrogenicity of a tamoxifen analog. 1995 Aug 2