Raloxifene Hydrochloride

estrogen receptor 1 ; Homo sapiens







166 Article(s)
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1 34404919 Repurposing the estrogen receptor modulator raloxifene to treat SARS-CoV-2 infection. 2022 Jan 2
2 35007301 SERMs (selective estrogen receptor modulator), acting as estrogen receptor β agonists in hepatocellular carcinoma cells, inhibit the transforming growth factor-α-induced migration via specific inhibition of AKT signaling pathway. 2022 2
3 35286219 Mitophagy induction and aryl hydrocarbon receptor-mediated redox signaling contribute to the suppression of breast cancer cell growth by raloxifene via regulation of inflammasomes activation. 2022 Mar 14 5
4 35614039 Characterization of raloxifene as a potential pharmacological agent against SARS-CoV-2 and its variants. 2022 May 25 2
5 32940862 Raloxifene inhibits pancreatic adenocarcinoma growth by interfering with ERβ and IL-6/gp130/STAT3 signaling. 2021 Feb 3
6 33882282 Endocrine prevention of breast cancer. 2021 Jun 15 1
7 34319769 Breast Cancer Prevention: Time for Change. 2021 Dec 2
8 34398352 Turning scientific serendipity into discoveries in breast cancer research and treatment: a tale of PhD students and a 50-year roaming tamoxifen team. 2021 Nov 1
9 34509864 Benzothiophene derivatives as selective estrogen receptor covalent antagonists: Design, synthesis and anti-ERα activities. 2021 Oct 1 1
10 34572301 Raloxifene Ameliorates Glucosamine-Induced Insulin Resistance in Ovariectomized Rats. 2021 Aug 30 2
11 34630393 Sex Hormones and Aging Modulate Interferon Lambda 1 Production and Signaling by Human Uterine Epithelial Cells and Fibroblasts. 2021 2
12 32068570 Do we need sex-oriented clinical practice guidelines for the treatment of schizophrenia? 2020 May 1
13 32482672 Identification of Estrogen Receptor Modulators as Inhibitors of Flavivirus Infection. 2020 Jul 22 1
14 32656689 Chitosan-Raloxifene nanoparticle containing doxorubicin as a new double-effect targeting vehicle for breast cancer therapy. 2020 Dec 2
15 32871847 Raloxifene and Bazedoxifene Could Be Promising Candidates for Preventing the COVID-19 Related Cytokine Storm, ARDS and Mortality. 2020 Sep-Oct 1
16 33033707 An Overview of Cancer Prevention: Chemoprevention and Immunoprevention. 2020 Sep 30 1
17 33066585 Raloxifene as Treatment for Various Types of Brain Injuries and Neurodegenerative Diseases: A Good Start. 2020 Oct 14 2
18 31073029 The selective estrogen receptor modulator raloxifene mitigates the effect of all-trans-retinal toxicity in photoreceptor degeneration. 2019 Jun 14 1
19 31494144 Breast cancer chemoprevention: An update on current practice and opportunities for primary care physicians. 2019 Dec 1
20 28859903 Bazedoxifene and raloxifene protect neocortical neurons undergoing hypoxia via targeting ERα and PPAR-γ. 2018 Feb 5 1
21 28924735 The G protein-coupled estrogen receptor (GPER/GPR30) may serve as a prognostic marker in early-stage cervical cancer. 2018 Jan 1
22 29482944 Synthesis and biological evaluation of 4,6-diaryl-2-pyrimidinamine derivatives as anti-breast cancer agents. 2018 Apr 1 1
23 30241506 The estrogen receptor 1 gene affects bone mineral density and osteoporosis treatment efficiency in Slovak postmenopausal women. 2018 Sep 21 1
24 28396978 A Novel Strategy to Co-target Estrogen Receptor and Nuclear Factor κB Pathways with Hybrid Drugs for Breast Cancer Therapy. 2017 Jun 1
25 26133657 Effect of selective estrogen receptor modulators on metabolic homeostasis. 2016 May 1
26 26648459 A novel curcumin derivative increases the cytotoxicity of raloxifene in estrogen receptor-negative breast cancer cell lines. 2016 Jan 3
27 27185013 Synthesis and evaluation of raloxifene derivatives as a selective estrogen receptor down-regulator. 2016 Jul 1 1
28 27203377 Controlling Sulfuryl-Transfer Biology. 2016 May 19 3
29 27546373 Pharmacogenetic study of the effects of raloxifene on negative symptoms of postmenopausal women with schizophrenia: A double-blind, randomized, placebo-controlled trial. 2016 Oct 1
30 27576059 Daidzein increases OPG/RANKL ratio and suppresses IL-6 in MG-63 osteoblast cells. 2016 Nov 1
31 27842943 Raloxifene increases prefrontal activity during emotional inhibition in schizophrenia based on estrogen receptor genotype. 2016 Dec 5
32 28003814 The Selective Estrogen Receptor Modulator Raloxifene Inhibits Neutrophil Extracellular Trap Formation. 2016 1
33 25410727 In vitro evaluation of a tetrahydroisoquinoline derivative as a steroid sulfatase inhibitor and a selective estrogen receptor modulator. 2015 Feb 1
34 25537862 Raloxifene induces autophagy-dependent cell death in breast cancer cells via the activation of AMP-activated protein kinase. 2015 3
35 25795461 Induction of UDP-glucuronosyltransferase 2B15 gene expression by the major active metabolites of tamoxifen, 4-hydroxytamoxifen and endoxifen, in breast cancer cells. 2015 Jun 1
36 26289836 Selective estrogen receptor modulators and the combination therapy conjugated estrogens/bazedoxifene: A review of effects on the breast. 2015 Sep 3
37 26529585 Reversal effects of Raloxifene on paclitaxel resistance in 2 MDR breast cancer cells. 2015 3
38 23727128 Alzheimer's disease: review of hormone therapy trials and implications for treatment and prevention after menopause. 2014 Jul 1
39 24481452 The aryl hydrocarbon receptor mediates raloxifene-induced apoptosis in estrogen receptor-negative hepatoma and breast cancer cells. 2014 Jan 30 5
40 24498137 Elevated MiR-222-3p promotes proliferation and invasion of endometrial carcinoma via targeting ERα. 2014 1
41 24785473 Oestrogen induced downregulation of TFPI expression is mediated by ERα. 2014 Jul 1
42 24829621 Advances in Preventive Therapy for Estrogen-Receptor-Negative Breast Cancer. 2014 2
43 24930824 Acquired resistance to selective estrogen receptor modulators (SERMs) in clinical practice (tamoxifen & raloxifene) by selection pressure in breast cancer cell populations. 2014 Nov 1
44 25084324 From empirical to mechanism-based discovery of clinically useful Selective Estrogen Receptor Modulators (SERMs). 2014 Nov 2
45 25378950 Preventative therapies for healthy women at high risk of breast cancer. 2014 1
46 23613312 Design, synthesis, and biological evaluation of cyclopropyl analogues of stilbene with raloxifene side chain as subtype-selective ligands for estrogen receptor. 2013 Sep 1
47 23634843 Extranuclear ERα is associated with regression of T47D PKCα-overexpressing, tamoxifen-resistant breast cancer. 2013 May 1 3
48 23915737 Breast cancer prevention by antihormones and other drugs: where do we stand? 2013 Aug 2
49 24015958 The HER4 isoform JM-a/CYT2 relates to improved survival in bladder cancer patients but only if the estrogen receptor α is not expressed. 2013 Sep 2
50 24069582 Targeted therapy for breast cancer prevention. 2013 Sep 23 1