Amines

ETS transcription factor ERG ; Homo sapiens







10 Article(s)
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Title
Pub. Year
#Total Relationships
1 33521468 Spirocycle MmpL3 Inhibitors with Improved hERG and Cytotoxicity Profiles as Inhibitors of Mycobacterium tuberculosis Growth. 2021 Jan 26 1
2 29400967 Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design. 2018 Jul 26 1
3 26713112 Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety. 2015 Dec 10 1
4 24412109 Successful reduction of off-target hERG toxicity by structural modification of a T-type calcium channel blocker. 2014 Feb 1 1
5 21524576 2,6-Disubstituted pyrazines and related analogs as NR2B site antagonists of the NMDA receptor with anti-depressant activity. 2011 Jun 1 1
6 19914064 Synthesis and antiplasmodial activity of novel 2,4-diaminopyrimidines. 2010 Jan 1 1
7 18996007 The discovery of AZD5597, a potent imidazole pyrimidine amide CDK inhibitor suitable for intravenous dosing. 2008 Dec 15 1
8 17188866 Constrained 7-fluorocarboxychromone-4-aminopiperidine based Melanin-concentrating hormone receptor 1 antagonists: the effects of chirality on substituted indan-1-ylamines. 2007 Feb 15 1
9 17303420 The synthesis and biological evaluation of novel series of nitrile-containing fluoroquinolones as antibacterial agents. 2007 Apr 15 1
10 15566305 Potent N-(1,3-thiazol-2-yl)pyridin-2-amine vascular endothelial growth factor receptor tyrosine kinase inhibitors with excellent pharmacokinetics and low affinity for the hERG ion channel. 2004 Dec 2 1