bombesin-like receptor 3 ; Mus musculus






19 Article(s)
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1 12877936 Sibutramine sensitivity assay revealed a unique phenotype of bombesin BB3 receptor-deficient mice. Eur J Pharmacol 2003 Jul 18 1
2 15144894 Functions of pancreatic beta cells and adipocytes in bombesin receptor subtype-3-deficient mice. Biochem Biophys Res Commun 2004 Jun 4 3
3 18336841 Bombesin marine toxin conjugates inhibit the growth of lung cancer cells. Life Sci 2008 Apr 9 3
4 20219372 Synthesis and SAR of derivatives based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity. Bioorg Med Chem Lett 2010 Apr 1 3
5 20807840 Body temperature as a mouse pharmacodynamic response to bombesin receptor subtype-3 agonists and other potential obesity treatments. Am J Physiol Endocrinol Metab 2010 Nov 1
6 21036912 Antiobesity effect of MK-5046, a novel bombesin receptor subtype-3 agonist. J Pharmacol Exp Ther 2011 Feb 3
7 21878513 Bombesin receptor subtype-3 (BRS-3) regulates glucose-stimulated insulin secretion in pancreatic islets across multiple species. Endocrinology 2011 Nov 5
8 24412111 Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration. Bioorg Med Chem Lett 2014 Feb 1 1
9 24452453 Regulation of body temperature and brown adipose tissue thermogenesis by bombesin receptor subtype-3. Am J Physiol Endocrinol Metab 2014 Mar 1
10 24900253 Discovery of MK-5046, a Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity. ACS Med Chem Lett 2011 Jan 13 3
11 24900283 Discovery of benzodiazepine sulfonamide-based bombesin receptor subtype 3 agonists and their unusual chirality. ACS Med Chem Lett 2011 Dec 8 3
12 25497965 Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach. Bioorg Med Chem 2015 Jan 1 2
13 26801314 Bombesin-like receptor 3 regulates blood pressure and heart rate via a central sympathetic mechanism. Am J Physiol Heart Circ Physiol 2016 Apr 1 3
14 27491709 Synthesis and biological evaluation of novel imidazol-1-ylacetic acid derivatives as non-brain penetrant bombesin receptor subtype-3 (BRS-3) agonists. Bioorg Med Chem Lett 2016 Sep 1 2
15 29107299 Bombesin-like receptor 3 (Brs3) expression in glutamatergic, but not GABAergic, neurons is required for regulation of energy metabolism. Mol Metab 2017 Nov 1
16 31911345 Bombesin Receptor Subtype-3 in Human Diseases. Arch Med Res 2019 Oct 1
17 32229422 BRS3 in both MC4R- and SIM1-expressing neurons regulates energy homeostasis in mice. Mol Metab 2020 Jun 2
18 34038711 Preoptic BRS3 neurons increase body temperature and heart rate via multiple pathways. Cell Metab 2021 Jul 6 2
19 35405616 Discovery of oridonin as a novel agonist for BRS-3. Phytomedicine 2022 Jun 9