Title : Farnesyl Transferase Inhibitor Lonafarnib Enhances α7nAChR Expression Through Inhibiting DNA Methylation of CHRNA7 and Increases α7nAChR Membrane Trafficking.

Pub. Date : 2020

PMID : 33447242






1 Functional Relationships(s)
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1 Inhibition of Ras farnesylation in acute has been found to upregulate the alpha7 nicotinic acetylcholine receptor (alpha7nAChR) activity. Acetylcholine cholinergic receptor, nicotinic, alpha polypeptide 7 Mus musculus