Title : Tolerance to WIN55,212-2 is delayed in desensitization-resistant S426A/S430A mice.

Pub. Date : 2019 Apr

PMID : 30629988






2 Functional Relationships(s)
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Protein Name
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1 Mice expressing a mutant form of CB1, in which the serine residues at two putative phosphorylation sites necessary for desensitization have been replaced by non-phosphorylatable alanines (S426A/S430A), display reduced tolerance to Delta9-tetrahydrocannabinol (Delta9-THC). Dronabinol cannabinoid receptor 1 (brain) Mus musculus
2 Mice expressing a mutant form of CB1, in which the serine residues at two putative phosphorylation sites necessary for desensitization have been replaced by non-phosphorylatable alanines (S426A/S430A), display reduced tolerance to Delta9-tetrahydrocannabinol (Delta9-THC). Dronabinol cannabinoid receptor 1 (brain) Mus musculus