Title : Covalent inhibition of histone deacetylase 8 by 3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazin-6-imine.

Pub. Date : 2019 Mar

PMID : 30611847






1 Functional Relationships(s)
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Sentence
Compound Name
Protein Name
Organism
1 Further optimization of non-covalent interaction and thiol-reactivity provides opportunities to develop therapeutic useful covalent HDAC8 inhibitors. Sulfhydryl Compounds histone deacetylase 8 Homo sapiens