Title : MALT1 Inhibition Is Efficacious in Both Naïve and Ibrutinib-Resistant Chronic Lymphocytic Leukemia.

Pub. Date : 2017 Dec 15

PMID : 28993409






1 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 The ibrutinib target, Bruton"s tyrosine kinase (BTK), is essential for B-cell receptor signaling, and most resistant cases carry mutations in BTK or PLCG2, a downstream effector target of BTK. ibrutinib phospholipase C gamma 2 Homo sapiens