Title : Ketoconazole increases plasma concentrations of antimalarial mefloquine in healthy human volunteers.

Pub. Date : 2005 Jun

PMID : 15896247






2 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 The major metabolite of quinine is 3-hydroxyquinine formed by cytochrome P450 3A4 (CYP3A4). Quinine cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Ketoconazole, a potent inhibitor of CYP3A4, is known to markedly increase plasma concentrations of various co-administered drugs including quinine. Quinine cytochrome P450 family 3 subfamily A member 4 Homo sapiens