8-Hydroxy-2-(di-n-propylamino)tetralin

5-hydroxytryptamine receptor 1A ; Homo sapiens







293 Article(s)
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201 8021490 Inhibitors of serotonin synthesis and antagonists of serotonin 1A receptors inhibit T lymphocyte function in vitro and cell-mediated immunity in vivo. 1994 Jul 15 1
202 8138923 Agonist-induced desensitization and loss of high-affinity binding sites of stably expressed human 5-HT1A receptors. 1994 Mar 1
203 8199864 Modulation of light-induced C-Fos expression in the suprachiasmatic nuclei by 5-HT1A receptor agonists. 1994 Feb 28 2
204 8199879 Quantitative autoradiography of 5-HT1D and 5-HT1E binding sites labelled by [3H]5-HT, in frontal cortex and the hippocampal region of the human brain. 1994 Feb 28 1
205 8200427 Effect of activation of 5-HT1A receptors at the ventral medulla on phrenic nerve activity. 1994 Mar 3 2
206 8301575 Novel benzodioxopiperazines acting as antagonists at postsynaptic 5-HT1A receptors and as agonists at 5-HT1A autoreceptors: a comparative pharmacological characterization with proposed 5-HT1A antagonists. 1994 Jan 2
207 7680787 The presence of a serotonin uptake inhibitor alters pharmacological manipulations of serotonin release. 1993 Jan 2
208 7870936 Serotonin involvement in the discriminative stimulus effects of kappa opioids in pigeons. 1993 1
209 8005619 Role of lipids in receptor mediated signal transduction. 1993 Dec 1
210 8098761 In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol. 1993 May 1
211 8101137 Lateral tegmental field involvement in the central sympathoinhibitory action of 8-OH-DPAT. 1993 May 28 1
212 8381359 S 15535: a highly selective benzodioxopiperazine 5-HT1A receptor ligand which acts as an agonist and an antagonist at presynaptic and postsynaptic sites respectively. 1993 Jan 5 1
213 8382063 Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cells. 1993 Jan 26 1
214 8389958 Serotonin modulates the levels of mRNAS coding for thyrotropin-releasing hormone and preprotachykinin by different mechanisms in medullary raphe neurons. 1993 Mar 2
215 8430834 Immunohistochemical mapping of cellular and subcellular distribution of 5-HT1A receptors in rat and human kidneys. 1993 Jan 2
216 8459396 Centrally acting serotonergic agents. Synthesis and structure-activity relationships of C-1- or C-3-substituted derivatives of 8-hydroxy-2-(di-n-propylamino)tetralin. 1993 Mar 19 1
217 8461029 Characterization of recombinant human serotonin 5HT1A receptors expressed in Chinese hamster ovary cells. [3H]spiperone discriminates between the G-protein-coupled and -uncoupled forms. 1993 Mar 9 1
218 8490207 Serotonin and the mammalian circadian system: I. In vitro phase shifts by serotonergic agonists and antagonists. 1993 Spring 1
219 8497336 Antidepressant-like activity of compounds with varying efficacy at 5-HT1A receptors. 1993 Apr 1
220 1316283 Effects of 5-HT1A receptor agonists on the circadian rhythm of wheel-running activity in hamsters. 1992 Apr 7 1
221 1318516 Mediation of serotonin hyperalgesia by the cAMP second messenger system. 1992 1
222 1356248 The effects of pertussis toxin on dopamine D2 and serotonin 5-HT1A autoreceptor-mediated inhibition of neurotransmitter synthesis: relationship to receptor reserve. 1992 May 2
223 1357094 Characterization of the 5-hydroxytryptamine receptor modulating the release of 5-[3H]hydroxytryptamine in slices of the human neocortex. 1992 Oct 1
224 1387027 Evidence for postsynaptic mediation of the hypothermic effect of 5-HT1A receptor activation. 1992 Jul 1
225 1389001 Citalopram and 8-OH-DPAT attenuate nicotine-induced excitation of central noradrenaline neurons. 1992 1
226 1409788 The 5-HT1A agonist 8-OH-DPAT attenuates the satiating action of cholecystokinin. 1992 Jul 1
227 1410132 Role of spinal serotonin1 receptor subtypes in thermally and mechanically elicited nociceptive reflexes. 1992 1
228 1426017 Clozapine has sub-micromolar affinity for 5-HT1A receptors in human brain tissue. 1992 Oct 20 1
229 1436121 Differential coupling of 5-HT1A receptors occupied by 5-HT or 8-OH-DPAT to adenylyl cyclase. 1992 Oct 1
230 1436390 Desensitization of 5-HT1A autoreceptors by chronic administration of 8-OH-DPAT. 1992 Oct 3
231 1446239 The physiological effects of serotonin are mediated by the 5HT1A receptor in the cat's cerebellar cortex. 1992 Sep 25 1
232 1448178 Functional expression of human 5-HT1A receptors and differential coupling to second messengers in CHO cells. 1992 Aug 2
233 1468487 (-)-Penbutolol as a blocker of central 5-HT1A receptor-mediated responses. 1992 Nov 3 2
234 1531359 Antagonism studies with BMY-7378 and NAN-190: effects on 8-hydroxy-2-(di-n-propylamino)tetralin-induced increases in punished responding of pigeons. 1992 Feb 1
235 1535691 Agonist/antagonist interactions with cloned human 5-HT1A receptors: variations in intrinsic activity studied in transfected HeLa cells. 1992 Mar 1
236 1658007 Actions of 8-hydroxy-2-(N-dipropylamino) tetralin (8-OH-DPAT) at alpha 2-adrenoceptors. 1991 Aug 1
237 1664803 Contractile effects of 8-hydroxy-2-(di-n-propylamino)tetralin and flesinoxan in human isolated basilar artery. 1991 Sep 4 3
238 1667606 Autoradiographic distribution of alpha 2 adrenoceptors, NAIBS, and 5-HT1A receptors in human brain using [3H]idazoxan and [3H]rauwolscine. 1991 Dec 6 1
239 1683291 Sympatholytic action of yohimbine mediated by 5-HT1A receptors. 1991 Jun 25 2
240 1715390 Extracellular serotonin levels change with behavioral state but not with pyrogen-induced hyperthermia. 1991 Sep 1
241 1762063 Imipramine as a discriminative stimulus. 1991 Dec 1
242 1772068 Serotonin: its role and receptors in enteric neurotransmission. 1991 1
243 1819150 Central 5-hydroxytryptamine (5-HT) receptors in blood pressure regulation. 1991 Nov-Dec 1
244 1824956 Increase in serotonin 5-HT1A receptors in prefrontal and temporal cortices of brains from patients with chronic schizophrenia. 1991 1
245 1825686 Antagonism by 8-hydroxy-2(di-n-propylamino)tetraline and other serotonin agonists of muscarinic M1-type receptors coupled to inositol phospholipid breakdown in human IMR-32 and SK-N-MC neuroblastoma cells. 1991 1
246 1828519 Antidepressant-like effects of buspirone mediated by the 5-HT1A post-synaptic receptors in the learned helplessness paradigm. 1991 1
247 1829231 Involvement of 5-HT1A activity in the discriminative stimulus effects of imipramine. 1991 Feb 1
248 1834090 Serotonergic measures in suicide brain: 5-HT1A binding sites in frontal cortex of suicide victims. 1991 1
249 1834306 Autoradiographic analysis of serotonin 5-HT1A receptor binding in the human brain postmortem: effects of age and alcohol. 1991 Jul 19 1
250 1838579 Characterization of 5-hydroxytryptamine 1A-like binding sites in human ganglioneuroblastoma. 1991 Oct 28 1