1 Article(s)Download |
PMID | Title | Pub. Year | #Total Relationships |
1 | 22517972 | Sequential metabolism of AMG 487, a novel CXCR3 antagonist, results in formation of quinone reactive metabolites that covalently modify CYP3A4 Cys239 and cause time-dependent inhibition of the enzyme. | 2012 Jul | 1 |