| 1 |
32531951 | Androgen Deprivation Induces Reprogramming of Prostate Cancer Cells to Stem-Like Cells. | 2020 Jun 10 |
1 |
| 2 |
30615932 | Halogen-substituted anthranilic acid derivatives provide a novel chemical platform for androgen receptor antagonists. | 2019 Apr |
3 |
| 3 |
31470108 | Androgen receptor activation reduces the endothelial cell proliferation through activating the cSrc/AKT/p38/ERK/NFκB-mediated pathway. | 2019 Nov |
2 |
| 4 |
29392883 | In silico binding of 4,4'-bisphenols predicts in vitro estrogenic and antiandrogenic activity. | 2018 May |
1 |
| 5 |
29720561 | Androgen Receptor Signaling Reduces Radiosensitivity in Bladder Cancer. | 2018 Jul |
1 |
| 6 |
28163245 | Anti-androgen 2-hydroxyflutamide modulates cadherin, catenin and androgen receptor phosphorylation in androgen-sensitive LNCaP and androgen-independent PC3 prostate cancer cell lines acting via PI3K/Akt and MAPK/ERK1/2 pathways. | 2017 Apr |
2 |
| 7 |
28711501 | Comparing the androgenic and estrogenic properties of progestins used in contraception and hormone therapy. | 2017 Sep 9 |
1 |
| 8 |
28832499 | A Molecular Modeling Study of the Hydroxyflutamide Resistance Mechanism Induced by Androgen Receptor Mutations. | 2017 Aug 23 |
5 |
| 9 |
26614265 | Hyperandrogenism Decreases GRP78 Protein Level and Glucose Uptake in Human Endometrial Stromal Cells. | 2016 Jun |
1 |
| 10 |
26813233 | Functional analysis of androgen receptor mutations that confer anti-androgen resistance identified in circulating cell-free DNA from prostate cancer patients. | 2016 Jan 26 |
1 |
| 11 |
26265743 | A Screen of Approved Drugs Identifies the Androgen Receptor Antagonist Flutamide and Its Pharmacologically Active Metabolite 2-Hydroxy-Flutamide as Heterotropic Activators of Cytochrome P450 3A In Vitro and In Vivo. | 2015 Nov |
1 |
| 12 |
23436650 | The discovery of novel human androgen receptor antagonist chemotypes using a combined pharmacophore screening procedure. | 2013 Apr |
1 |
| 13 |
23462715 | Development of silicon-containing bis-phenol derivatives as androgen receptor antagonists: selectivity switching by C/Si exchange. | 2013 Apr 1 |
1 |
| 14 |
23889773 | Amyloid precursor protein in human breast cancer: an androgen-induced gene associated with cell proliferation. | 2013 Nov |
1 |
| 15 |
24065547 | Testosterone promotes vascular endothelial cell migration via upregulation of ROCK-2/moesin cascade. | 2013 Dec |
2 |
| 16 |
22496481 | Identification and characterization of MEL-3, a novel AR antagonist that suppresses prostate cancer cell growth. | 2012 Jun |
4 |
| 17 |
22522230 | Does 2-hydroxyflutamide inhibit apoptosis in porcine granulosa cells? - An in vitro study. | 2012 |
2 |
| 18 |
22746350 | Design, synthesis, and biological evaluation of nonsteroidal cycloalkane[d]isoxazole-containing androgen receptor modulators. | 2012 Jul 26 |
1 |
| 19 |
22922989 | Epidermal growth factor induces bladder cancer cell proliferation through activation of the androgen receptor. | 2012 Nov |
2 |
| 20 |
21243325 | Hydroxyflutamide enhances cellular sensitivity to 5-fluorouracil by suppressing thymidylate synthase expression in bicalutamide-resistant human prostate cancer cells. | 2011 Mar |
1 |
| 21 |
21748440 | Androgen receptor coregulators NOCR1, TIF2, and ARA70 may account for the hydroxyflutamide insensitivity of prostate cancer cells. | 2011 Dec |
2 |
| 22 |
21796530 | Detection of ligand-selective interactions of the human androgen receptor by SELDI-MS-TOF. | 2011 |
2 |
| 23 |
21829708 | Modulation of androgen receptor signaling in hormonal therapy-resistant prostate cancer cell lines. | 2011 |
5 |
| 24 |
19787772 | Study of the impact of the T877A mutation on ligand-induced helix-12 positioning of the androgen receptor resulted in design and synthesis of novel antiandrogens. | 2010 Feb 15 |
1 |
| 25 |
20521823 | Design and synthesis of androgen receptor full antagonists bearing a p-carborane cage: promising ligands for anti-androgen withdrawal syndrome. | 2010 Jul 8 |
1 |
| 26 |
18548383 | Levonorgestrel antagonism on estrogen-induced pituitary tumors is mediated by progesterone receptors. | 2008 Apr |
1 |
| 27 |
18571420 | 4-(Anilino)pyrrole-2-carboxamides: Novel non-steroidal/non-anilide type androgen antagonists effective upon human prostate tumor LNCaP cells with mutated nuclear androgen receptor. | 2008 Jul 15 |
1 |
| 28 |
18596614 | Nandrolone decreases mu opioid receptor expression in SH-SY5Y human neuroblastoma cells. | 2008 Jul 16 |
1 |
| 29 |
17223690 | The androgen receptor T877A mutant recruits LXXLL and FXXLF peptides differently than wild-type androgen receptor in a time-resolved fluorescence resonance energy transfer assay. | 2007 Jan 23 |
1 |
| 30 |
17541168 | Dihydrotestosterone inhibits tumor necrosis factor alpha induced interleukin-1alpha mRNA expression in rheumatoid fibroblast-like synovial cells. | 2007 Jun |
1 |
| 31 |
17553795 | Glyceraldehyde-3-phosphate dehydrogenase enhances transcriptional activity of androgen receptor in prostate cancer cells. | 2007 Aug 3 |
1 |
| 32 |
17587566 | PRMT2, a member of the protein arginine methyltransferase family, is a coactivator of the androgen receptor. | 2007 Oct |
2 |
| 33 |
17636177 | Testosterone inhibits matrix metalloproteinase-1 production in human endometrial stromal cells in vitro. | 2007 Jun |
1 |
| 34 |
17656415 | Human sperm express a functional androgen receptor: effects on PI3K/AKT pathway. | 2007 Oct |
2 |
| 35 |
17073766 | Mechanisms of androgen receptor repression in prostate cancer. | 2006 Dec |
1 |
| 36 |
15538745 | 5alpha-dihydrotestosterone inhibits 1alpha,25-dihydroxyvitamin D3-induced expression of CYP24 in human prostate cancer cells. | 2005 May 15 |
2 |
| 37 |
15900601 | Androgen receptor modifications in prostate cancer cells upon long-termandrogen ablation and antiandrogen treatment. | 2005 Nov 1 |
1 |
| 38 |
15994236 | The structural basis of androgen receptor activation: intramolecular and intermolecular amino-carboxy interactions. | 2005 Jul 12 |
1 |
| 39 |
16054371 | Prostate cancer PET bioprobes: synthesis of [18F]-radiolabeled hydroxyflutamide derivatives. | 2005 Nov 15 |
1 |
| 40 |
16129672 | Structural basis for accommodation of nonsteroidal ligands in the androgen receptor. | 2005 Nov 11 |
3 |
| 41 |
14593076 | Antiandrogen effects of mifepristone on coactivator and corepressor interactions with the androgen receptor. | 2004 Jan |
1 |
| 42 |
14973257 | Interactions between androgen and growth factors in granulosa cell subtypes of porcine antral follicles. | 2004 Jul |
1 |
| 43 |
15219414 | Oxandrolone blocks glucocorticoid signaling in an androgen receptor-dependent manner. | 2004 May |
2 |
| 44 |
12672951 | 3 beta-acetoxyandrost-1,5-diene-17-ethylene ketal functions as a potent antiandrogen with marginal agonist activity. | 2003 Apr 15 |
1 |
| 45 |
11916967 | Liganded androgen receptor interaction with beta-catenin: nuclear co-localization and modulation of transcriptional activity in neuronal cells. | 2002 Jun 7 |
1 |
| 46 |
12114440 | Acquisition of agonistic properties of nonsteroidal antiandrogens after treatment with oncostatin M in prostate cancer cells. | 2002 Jul |
2 |
| 47 |
12123801 | Pure antiandrogens disrupt the recruitment of coactivator GRIP1 to colocalize with androgen receptor in nuclei. | 2002 Jul 17 |
1 |
| 48 |
12153751 | Regulation of osteoprotegerin production by androgens and anti-androgens in human osteoblastic lineage cells. | 2002 Aug |
2 |
| 49 |
12573819 | Antiandrogens: selective androgen receptor modulators. | 2002 Dec 30 |
1 |
| 50 |
12573820 | Potential action of IGF-1 and EGF on androgen receptor nuclear transfer and transactivation in normal and cancer human prostate cell lines. | 2002 Dec 30 |
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