Crizotinib

ATP-binding cassette, sub-family B (MDR/TAP), member 1B ; Mus musculus







3 Article(s)
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1 26361725 Brain accumulation of the EML4-ALK inhibitor ceritinib is restricted by P-glycoprotein (P-GP/ABCB1) and breast cancer resistance protein (BCRP/ABCG2). 2015 Dec 1
2 24037730 Increased oral availability and brain accumulation of the ALK inhibitor crizotinib by coadministration of the P-glycoprotein (ABCB1) and breast cancer resistance protein (ABCG2) inhibitor elacridar. 2014 Mar 15 2
3 22233293 Crizotinib (PF-02341066) reverses multidrug resistance in cancer cells by inhibiting the function of P-glycoprotein. 2012 Jul 6