| 1 |
35328343 | Chemical Synthesis, Pharmacokinetic Properties and Biological Effects of JM-00266, a Putative Non-Brain Penetrant Cannabinoid Receptor 1 Inverse Agonist. | 2022 Mar 8 |
1 |
| 2 |
33931733 | Cannabinoid receptor activation acutely increases synaptic vesicle numbers by activating synapsins in human synapses. | 2021 Nov |
1 |
| 3 |
32101383 | Differential activation of G protein-mediated signaling by synthetic cannabinoid receptor agonists. | 2020 Apr |
2 |
| 4 |
32702414 | Translation of in vitro cannabinoid 1 receptor agonist activity to in vivo pharmacodynamic endpoints. | 2020 Jul - Aug |
1 |
| 5 |
33002729 | Chlorotrimethylsilane promoted one-flask heterocyclic synthesis of 1,2,4-triazoles from nitrilimines: Modeling studies and bioactivity evaluation of LH-21 and Rimonabant analogues. | 2020 Nov |
1 |
| 6 |
30636986 | 5F-Cumyl-PINACA in 'e-liquids' for electronic cigarettes: comprehensive characterization of a new type of synthetic cannabinoid in a trendy product including investigations on the in vitro and in vivo phase I metabolism of 5F-Cumyl-PINACA and its non-fluorinated analog Cumyl-PINACA. | 2019 |
1 |
| 7 |
29187590 | Selective Cannabinoid 2 Receptor Stimulation Reduces Tubular Epithelial Cell Damage after Renal Ischemia-Reperfusion Injury. | 2018 Feb |
1 |
| 8 |
29662438 | Cannabinoid Receptor Type 1 Expression in the Developing Avian Retina: Morphological and Functional Correlation With the Dopaminergic System. | 2018 |
3 |
| 9 |
27504870 | Phase I metabolism of the highly potent synthetic cannabinoid MDMB-CHMICA and detection in human urine samples. | 2017 May |
1 |
| 10 |
27989582 | Expression of Cannabinoid Type 1 Receptors in Human Odontoblast Cells. | 2017 Feb |
1 |
| 11 |
28445587 | CB1 receptors down-regulate a cAMP/Epac2/PLC pathway to silence the nerve terminals of cerebellar granule cells. | 2017 Aug |
2 |
| 12 |
28516479 | Gαs signalling of the CB1 receptor and the influence of receptor number. | 2017 Aug |
2 |
| 13 |
28750814 | Real-Time Measurement of Cannabinoid Receptor-Mediated cAMP Signaling. | 2017 |
1 |
| 14 |
28861508 | Affinity and Efficacy Studies of Tetrahydrocannabinolic Acid A at Cannabinoid Receptor Types One and Two. | 2017 |
1 |
| 15 |
29161035 | Synthesis of Photoswitchable Δ9-Tetrahydrocannabinol Derivatives Enables Optical Control of Cannabinoid Receptor 1 Signaling. | 2017 Dec 20 |
1 |
| 16 |
27046127 | Mapping Cannabinoid 1 Receptor Allosteric Site(s): Critical Molecular Determinant and Signaling Profile of GAT100, a Novel, Potent, and Irreversibly Binding Probe. | 2016 Jun 15 |
1 |
| 17 |
27115025 | Optimization of cAMP fluorescence dataset from ACTOne cannabinoid receptor 1 cell line. | 2016 Jun |
1 |
| 18 |
27260125 | Pharmacological characterization of emerging synthetic cannabinoids in HEK293T cells and hippocampal neurons. | 2016 Sep 5 |
1 |
| 19 |
27506997 | Cannabinoid-induced depression of synaptic transmission is switched to stimulation when dopaminergic tone is increased in the globus pallidus of the rodent. | 2016 Nov |
1 |
| 20 |
28066250 | Selective Estrogen Receptor Modulators: Cannabinoid Receptor Inverse Agonists with Differential CB1 and CB2 Selectivity. | 2016 |
1 |
| 21 |
25978068 | Molecular-interaction and signaling profiles of AM3677, a novel covalent agonist selective for the cannabinoid 1 receptor. | 2015 Aug 19 |
1 |
| 22 |
26203658 | Distinct Temporal Fingerprint for Cyclic Adenosine Monophosphate (cAMP) Signaling of Indole-2-carboxamides as Allosteric Modulators of the Cannabinoid Receptors. | 2015 Aug 13 |
2 |
| 23 |
24264530 | Delineation of domains within the cannabinoid CB1 and dopamine D2 receptors that mediate the formation of the heterodimer complex. | 2014 May |
4 |
| 24 |
24533119 | Cannabinoid type 1 receptors transiently silence glutamatergic nerve terminals of cultured cerebellar granule cells. | 2014 |
1 |
| 25 |
25154875 | Peripheral cannabinoid 1 receptor blockade activates brown adipose tissue and diminishes dyslipidemia and obesity. | 2014 Dec |
1 |
| 26 |
23667597 | The second intracellular loop of the human cannabinoid CB2 receptor governs G protein coupling in coordination with the carboxyl terminal domain. | 2013 |
1 |
| 27 |
24148245 | CB1 and CB2 receptors are novel molecular targets for Tamoxifen and 4OH-Tamoxifen. | 2013 Nov 15 |
1 |
| 28 |
22482014 | Endocannabinoid-binding CB1 and TRPV1 receptors as modulators of sperm capacitation. | 2012 Jan 1 |
2 |
| 29 |
22823387 | Expression and functions of μ-opioid receptors and cannabinoid receptors type 1 in T lymphocytes. | 2012 Jul |
1 |
| 30 |
21216016 | Inverse agonism of cannabinoid CB1 receptor blocks the adhesion of encephalitogenic T cells in inflamed brain venules by a protein kinase A-dependent mechanism. | 2011 Apr |
1 |
| 31 |
21781118 | Δ9-THC increases endogenous AHA1 expression in rat cerebellum and may modulate CB1 receptor function during chronic use. | 2011 Sep |
1 |
| 32 |
21829686 | Type-1 cannabinoid receptors reduce membrane fluidity of capacitated boar sperm by impairing their activation by bicarbonate. | 2011 |
2 |
| 33 |
24900275 | Identification of a Potent and Selective Cannabinoid CB1 Receptor Antagonist from Auxarthron reticulatum. | 2011 Nov 10 |
1 |
| 34 |
19818494 | L-type channel inhibition by CB1 cannabinoid receptors is mediated by PTX-sensitive G proteins and cAMP/PKA in GT1-7 hypothalamic neurons. | 2009 Nov-Dec |
2 |
| 35 |
19858202 | Cannabinoid receptor type 1- and 2-mediated increase in cyclic AMP inhibits T cell receptor-triggered signaling. | 2009 Dec 18 |
2 |
| 36 |
17686497 | Regulation of DARPP-32 phosphorylation by Delta9-tetrahydrocannabinol. | 2008 Jan |
1 |
| 37 |
18156315 | Analysis of promoter regions regulating basal and interleukin-4-inducible expression of the human CB1 receptor gene in T lymphocytes. | 2008 Mar |
1 |
| 38 |
18566465 | Cannabinoid receptors in conjunctival epithelium: identification and functional properties. | 2008 Oct |
1 |
| 39 |
16395612 | Presence of the cannabinoid receptors, CB1 and CB2, in human omental and subcutaneous adipocytes. | 2006 Aug |
2 |
| 40 |
16690806 | FOXO1A differentially regulates genes of decidualization. | 2006 Aug |
1 |
| 41 |
16893424 | Cannabinoid receptors in human astroglial tumors. | 2006 Aug |
1 |
| 42 |
16953186 | In vitro and in vivo pharmacology of synthetic olivetol- or resorcinol-derived cannabinoid receptor ligands. | 2006 Oct |
1 |
| 43 |
16083441 | Purification and mass spectroscopic analysis of human CB1 cannabinoid receptor functionally expressed using the baculovirus system. | 2005 Sep |
2 |
| 44 |
16279794 | Design, synthesis, and binding studies of new potent ligands of cannabinoid receptors. | 2005 Nov 17 |
1 |
| 45 |
12737320 | Dual effect of cannabinoid CB1 receptor stimulation on a vanilloid VR1 receptor-mediated response. | 2003 Mar |
2 |
| 46 |
12759440 | Subversion and utilization of the host cell cyclic adenosine 5'-monophosphate/protein kinase A pathway by Brucella during macrophage infection. | 2003 Jun 1 |
1 |
| 47 |
10188977 | Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656, and AM630. | 1999 Feb |
1 |
| 48 |
10217281 | Involvement of the carboxyl terminus of the third intracellular loop of the cannabinoid CB1 receptor in constitutive activation of Gs. | 1999 May |
4 |
| 49 |
10336536 | Synthesis and characterization of potent and selective agonists of the neuronal cannabinoid receptor (CB1). | 1999 Jun |
1 |
| 50 |
10422789 | Dual intracellular signaling pathways mediated by the human cannabinoid CB1 receptor. | 1999 Jun 25 |
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