Loperamide






179 Article(s)
Download
PMID
Title
Journal
Pub. Date
#Total Relationship(s)
1 1322429 Effects of loperamide on the human hypothalamo-pituitary-adrenal axis in vivo and in vitro. J Clin Endocrinol Metab 1992 Aug 5
2 2297461 Effect of increasing oral doses of loperamide on gallbladder motility in man. Br J Clin Pharmacol 1990 Jan 1
3 2545766 Effects of the opiate agonist loperamide on pituitary-adrenal function in patients with suspected hypercortisolism. J Endocrinol Invest 1989 Jan 4
4 2820051 Loperamide--an opiate receptor agonist with gastrointestinal motility effects. Scand J Gastroenterol Suppl 1987 1
5 2832297 Loperamide modifies but does not block the corticotropin-releasing hormone-induced ACTH response in patients with Addison's disease. Horm Metab Res Suppl 1987 5
6 2836258 Calmodulin-mediated effects of loperamide on chloride transport by brush border membrane vesicles from human ileum. Gastroenterology 1988 Jul 7
7 2855105 Loperamide, an opiate analog, differently modifies the adrenocorticotropin responses to corticotropin-releasing hormone and lysine vasopressin in patients with Addison's disease. Neuroendocrinology 1988 Dec 17
8 2901674 Evidence for a peripheral action of thyrotropin releasing hormone on gastrointestinal transit in mice. Neuropharmacology 1988 Apr 2
9 2979685 Effect of two potent calmodulin antagonists on calcium transport of brush border and basolateral vesicles from human duodenum. Aliment Pharmacol Ther 1987 Oct 2
10 3024866 Loperamide, an opiate analogue, inhibits plasma ACTH levels in patients with Addison's disease. Clin Endocrinol (Oxf) 1986 May 4
11 6319884 Loperamide: evidence of interaction with mu and delta opioid receptors. Life Sci 1983 1
12 6382576 Mechanisms of action of loperamide. Scand J Gastroenterol Suppl 1984 1
13 7544198 The anti-emetic effects of CP-99,994 in the ferret and the dog: role of the NK1 receptor. Br J Pharmacol 1995 May 1
14 7699214 Comparison between the suppressive effects of dexamethasone and loperamide on cortisol and ACTH secretion in some pathological conditions. J Endocrinol Invest 1994 Nov 1
15 8090278 In man the mu-opiate agonist loperamide specifically inhibits ACTH secretion induced by the cholecystokinin-like peptide ceruletide. Neuroendocrinology 1994 Jul 6
16 8232760 Loperamide inhibits corticotrophic cell function by a naloxone-insensitive mechanism in the rat in vitro. Neuroendocrinology 1993 Jun 2
17 8508715 Loperamide. Survey of studies on mechanism of its antidiarrheal activity. Dig Dis Sci 1993 Jun 1
18 8574143 Calmodulin inhibitors and calcium channel blockers influence dideoxycytidine renal excretion. Cell Mol Biol (Noisy-le-grand) 1995 2
19 8647944 P-glycoprotein in the blood-brain barrier of mice influences the brain penetration and pharmacological activity of many drugs. J Clin Invest 1996 Jun 1 4
20 8877029 Suppression of vagus-mediated pancreatic polypeptide release by the mu-opiate receptor agonist loperamide in man. Br J Clin Pharmacol 1996 Sep 6
21 9575405 [The delivery of loperamide to the brain by using polybutyl cyanoacrylate nanoparticles]. Eksp Klin Farmakol 1998 Jan-Feb 2
22 10717506 An overview of clinical studies with racecadotril in adults. Int J Antimicrob Agents 2000 Feb 1
23 10718373 Differential regulation of Ca2+ influx by fMLP and PAF in human neutrophils: possible involvement of store-operated Ca2+ channel. Shock 2000 Mar 2
24 10742982 Multidrug-resistance transporters. Pharm Biotechnol 1999 1
25 10766372 Determination of loperamide in rat plasma and bovine serum albumin by LC. J Pharm Biomed Anal 2000 Apr 1
26 10875545 Effect of loperamide on Na+/D-glucose cotransporter activity in mouse small intestine. J Pharm Pharmacol 2000 Jun 3
27 11474216 Effects of loperamide and other opioid-related substances on the transcriptional regulation of the rat pro-opiomelanocortin gene in AtT20 cells. Neuroendocrinology 2001 Aug 3
28 11939306 Frequency of the mutant MDR1 allele associated with ivermectin sensitivity in a sample population of collies from the northwestern United States. Am J Vet Res 2002 Apr 1
29 11964599 Interaction of morphine, fentanyl, sufentanil, alfentanil, and loperamide with the efflux drug transporter P-glycoprotein. Anesthesiology 2002 Apr 4
30 12164380 Apolipoprotein-mediated transport of nanoparticle-bound drugs across the blood-brain barrier. J Drug Target 2002 Jun 2
31 12948013 Quantitative evaluation of the function of small intestinal P-glycoprotein: comparative studies between in situ and in vitro. Pharm Res 2003 Aug 1
32 14516411 Loperamide increases glucose ultilization in streptozotocin-induced diabetic rats. Clin Exp Pharmacol Physiol 2003 Oct 4
33 14583678 Effects of ABCB1 (multidrug resistance transporter) gene mutations on disposition and central nervous effects of loperamide in healthy volunteers. Pharmacogenetics 2003 Nov 5
34 14586389 No effect of MDR1 C3435T variant on loperamide disposition and central nervous system effects. Clin Pharmacol Ther 2003 Nov 1
35 14613723 Potential roles of P-gp and calcium channels in loperamide and diphenoxylate transport. Toxicol Appl Pharmacol 2003 Nov 15 1
36 14765742 Loperamide toxicity in a collie with the MDR1 mutation associated with ivermectin sensitivity. J Vet Intern Med 2004 Jan-Feb 1
37 15244080 pH dependent uptake of loperamide across the gastrointestinal tract: an in vitro study. Drug Dev Ind Pharm 2004 May 7
38 15501934 The elementary mass action rate constants of P-gp transport for a confluent monolayer of MDCKII-hMDR1 cells. Biophys J 2005 Jan 4
39 15553234 Use of loperamide as a phenotypic probe of mdr1a status in CF-1 mice. Pharm Res 2004 Oct 1
40 15687373 Hydrolysis of capecitabine to 5'-deoxy-5-fluorocytidine by human carboxylesterases and inhibition by loperamide. J Pharmacol Exp Ther 2005 Jun 2
41 15835747 Relationship between loperamide-induced sedative effect and digoxin pharmacokinetics in healthy Japanese subjects. Pharm Res 2005 Mar 4
42 15942125 Loperamide inhibits tachykinin NK3-receptor-triggered serotonin release without affecting NK2-receptor-triggered serotonin release from guinea pig colonic mucosa. J Pharmacol Sci 2005 Jun 2
43 15959754 Activation of opioid mu-receptors by loperamide to improve interleukin-6-induced inhibition of insulin signals in myoblast C2C12 cells. Diabetologia 2005 Jul 2
44 16185316 mu-Opiate receptor agonist loperamide blocks bethanechol-induced gallbladder contraction, despite higher cholecystokinin plasma levels in man. Neurogastroenterol Motil 2005 Oct 8
45 16406665 Effect of opioid mu-receptors activation on insulin signals damaged by tumor necrosis factor alpha in myoblast C2C12 cells. Neurosci Lett 2006 Apr 24 2
46 16537797 Differential in vivo sensitivity to inhibition of P-glycoprotein located in lymphocytes, testes, and the blood-brain barrier. J Pharmacol Exp Ther 2006 Jun 1
47 16554356 Covalent linkage of apolipoprotein e to albumin nanoparticles strongly enhances drug transport into the brain. J Pharmacol Exp Ther 2006 Jun 1
48 17664252 Specificity of procaine and ester hydrolysis by human, minipig, and rat skin and liver. Drug Metab Dispos 2007 Nov 1
49 17683917 A review on the impact of P-glycoprotein on the penetration of drugs into the brain. Focus on psychotropic drugs. Eur Neuropsychopharmacol 2008 Mar 1
50 17889094 Hydrolysis of a series of parabens by skin microsomes and cytosol from human and minipigs and in whole skin in short-term culture. Toxicol Appl Pharmacol 2007 Dec 1 1