Title : FoxO1 regulates myocardial glucose oxidation rates via transcriptional control of pyruvate dehydrogenase kinase 4 expression.

Pub. Date : 2017 Sep 1

PMID : 28687587






2 Functional Relationships(s)
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1 Both pharmacological (1 microM AS1842856) and genetic (siRNA mediated) inhibition of FoxO1 decreased Pdk4/PDHK4 expression and subsequent PDH phosphorylation in H9c2 cardiac myocytes, whereas 10 microM dexamethasone-induced Pdk4/PDHK4 expression was abolished via pretreatment with 1 microM AS1842856. 5-amino-7-(cyclohexylamino)-1-ethyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid forkhead box O1 Mus musculus
2 Both pharmacological (1 microM AS1842856) and genetic (siRNA mediated) inhibition of FoxO1 decreased Pdk4/PDHK4 expression and subsequent PDH phosphorylation in H9c2 cardiac myocytes, whereas 10 microM dexamethasone-induced Pdk4/PDHK4 expression was abolished via pretreatment with 1 microM AS1842856. 5-amino-7-(cyclohexylamino)-1-ethyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid forkhead box O1 Mus musculus