Title : The activity of selective sigma-1 receptor ligands in seizure models in vivo.

Pub. Date : 2017 Jun 15

PMID : 28389336






1 Functional Relationships(s)
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1 Sig1R antagonist NE-100 at a dose of 25mg/kg demonstrated pro-convulsive activity on PTZ-induced seizures. N,N-dipropyl-2-(4-methoxy-3-(2-phenylethoxy)phenyl)ethylamine monohydrochloride sigma non-opioid intracellular receptor 1 Mus musculus