Pub. Date : 1992 Sep
PMID : 1324149
8 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
| 1 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | emodepside | endothelin receptor type A | Homo sapiens |
| 2 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | D-Tryptophan | endothelin receptor type A | Homo sapiens |
| 3 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | D-Aspartic acid | endothelin receptor type A | Homo sapiens |
| 4 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | L-Pro | endothelin receptor type A | Homo sapiens |
| 5 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | D-Valine | endothelin receptor type A | Homo sapiens |
| 6 | This was further confirmed by the use of a cyclic pentapeptide [cyclo(D-Trp,D-Asp,L-Pro, D-Val,L-Leu)] (BQ123), which is selective for ETA receptors. | Leucine | endothelin receptor type A | Homo sapiens |
| 7 | In the presence of 1 microM BQ123, [125I]ET-1 binding was decreased by 25-30%, whereas [125I]ET-3 binding was unaffected, confirming that 30-35% of ET receptors belong to the ETA subtypes, and that [125I]ET-1 bound to both ETA and ETB receptors with the same high affinity, but [125I]ET-3 bound only to ETB receptors with high affinity. | cyclo(Trp-Asp-Pro-Val-Leu) | endothelin receptor type A | Homo sapiens |
| 8 | In the presence of 1 microM BQ123, [125I]ET-1 binding was decreased by 25-30%, whereas [125I]ET-3 binding was unaffected, confirming that 30-35% of ET receptors belong to the ETA subtypes, and that [125I]ET-1 bound to both ETA and ETB receptors with the same high affinity, but [125I]ET-3 bound only to ETB receptors with high affinity. | cyclo(Trp-Asp-Pro-Val-Leu) | endothelin receptor type A | Homo sapiens |