Title : Macrolide antibacterials. Drug interactions of clinical significance.

Pub. Date : 1995 Aug

PMID : 7576262






1 Functional Relationships(s)
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1 Macrolide antibiotics can interact adversely with commonly used drugs, usually by altering metabolism due to complex formation and inhibition of cytochrome P-450 IIIA4 (CYP3A4) in the liver and enterocytes. macrolide antibiotics cytochrome P450 family 3 subfamily A member 4 Homo sapiens