Title : Effects of flavonols on P-glycoprotein activity in cultured rat hepatocytes.

Pub. Date : 1995

PMID : 7475916






1 Functional Relationships(s)
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1 In 72h-cultured hepatocytes, spontaneously overexpressing functional Pgp, flavonols inhibited R-123 efflux in a dose-dependent manner, but significantly reduced DOX retention while increasing its efflux. Doxorubicin ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus