Title : IRE-1-Targeting Caged Prodrug with Endoplasmic Reticulum Stress-Inducing and XBP-1S-Inhibiting Activities for Cancer Therapy.

Pub. Date : 2022 Apr 4

PMID : 35253431






1 Functional Relationships(s)
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1 Here, we report a novel prodrug, TC-D-F07, in which a thiol-reactive dinitrobenzenesulfonyl (Dns) cage was installed onto the C8 hydroxyl of the covalent IRE-1 inhibitor D-F07. 3,5-dinitrosalicylic acid endoplasmic reticulum to nucleus signaling 1 Homo sapiens