Title : Characterisation of bis(4-aminoquinoline)s as α1A adrenoceptor allosteric modulators.

Pub. Date : 2022 Feb 5

PMID : 34871559






1 Functional Relationships(s)
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1 A linear trend of increasing (3H)prazosin dissociation rate with increasing linker length between C7 and C11 was observed, confirming their action as allosteric modulators. Prazosin aldo-keto reductase family 1 member C4 Homo sapiens