Title : Exploring Ligand-Directed N-Acyl-N-alkylsulfonamide-Based Acylation Chemistry for Potential Targeted Degrader Development.

Pub. Date : 2021 Aug 12

PMID : 34413960






1 Functional Relationships(s)
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1 To test this possibility, we developed a series of CDK2-targeting N-acyl-N-alkylsulfonamide (NASA)-containing acylation probes. n-acyl-n-alkylsulfonamide cyclin dependent kinase 2 Homo sapiens