Title : Differences in P-glycoprotein activity in human and rodent blood-brain barrier assessed by mechanistic modelling.

Pub. Date : 2021 Sep

PMID : 34268580






2 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 BBB Pgp activity in the model was optimized using measured CSF data for the Pgp substrates ivermectin, indinavir, vincristine, docetaxel, paclitaxel, olanzapine and citalopram, as no useful in vitro data were available. Docetaxel ATP binding cassette subfamily B member 1 Homo sapiens
2 BBB Pgp activity in the model was optimized using measured CSF data for the Pgp substrates ivermectin, indinavir, vincristine, docetaxel, paclitaxel, olanzapine and citalopram, as no useful in vitro data were available. Docetaxel ATP binding cassette subfamily B member 1 Homo sapiens