Title : Effect of Genetic Variability in 20 Pharmacogenes on Concentrations of Tamoxifen and Its Metabolites.

Pub. Date : 2021 Jun 4

PMID : 34199712






1 Functional Relationships(s)
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1 BACKGROUND: Tamoxifen, as a treatment of estrogen receptor positive (ER+) breast cancer, is a weak anti-estrogen that requires metabolic activation to form metabolites with higher anti-estrogenic activity. Tamoxifen epiregulin Homo sapiens