Title : Cynandione A and PHA-543613 inhibit inflammation and stimulate macrophageal IL-10 expression following α7 nAChR activation.

Pub. Date : 2021 Aug

PMID : 33992630






1 Functional Relationships(s)
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1 Treatment with cynandione A and the specific alpha7 nicotinic acetylcholine receptor (alpha7 nAChR) agonist PHA-543613 remarkably reduced overexpression of proinflammatory cytokines, including tumor necrosis factor (TNF)-alpha, interleukin (IL)-6 and IL-1beta in lipopolysaccharide (LPS)-treated RAW264.7 cells and primary peritoneal macrophages, and endotoxemic mice. Acetylcholine cholinergic receptor, nicotinic, alpha polypeptide 7 Mus musculus