Title : ZYBT1, a potent, irreversible Bruton's Tyrosine Kinase (BTK) inhibitor that inhibits the C481S BTK with profound efficacy against arthritis and cancer.

Pub. Date : 2020 Aug

PMID : 32790160






2 Functional Relationships(s)
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1 ZYBT1 is a potent, irreversible, specific BTK inhibitor that inhibits the ibrutinib-resistant C481S BTK with nanomolar potency. ibrutinib Bruton agammaglobulinemia tyrosine kinase Mus musculus
2 ZYBT1 is a potent, irreversible, specific BTK inhibitor that inhibits the ibrutinib-resistant C481S BTK with nanomolar potency. ibrutinib Bruton agammaglobulinemia tyrosine kinase Mus musculus