Title : Potent Tetrahydroquinolone Eliminates Apicomplexan Parasites.

Pub. Date : 2020

PMID : 32626661






1 Functional Relationships(s)
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1 Herein, we create a next generation anti-apicomplexan lead compound, JAG21, a tetrahydroquinolone, with increased sp3-character to improve parasite selectivity. tetrahydroquinolinone Sp3 transcription factor Homo sapiens