Title : The β2-adrenoceptor agonist bronchodilators terbutaline and orciprenaline are also weak α1-adrenoceptor antagonists.

Pub. Date : 2020 Sep 5

PMID : 32592771






1 Functional Relationships(s)
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1 In conclusion, our work has provided additional quantitative evidence that terbutaline and orciprenaline are weak competitive alpha1-adrenoceptor antagonists, but this additional property is probably not therapeutically important in the clinical treatment of asthma or pulmonary artery hypertension with these more potent beta2-adrenoceptor agonists. Terbutaline adrenoceptor beta 2 Rattus norvegicus