Title : Slow-, Tight-Binding Inhibition of CYP17A1 by Abiraterone Redefines Its Kinetic Selectivity and Dosing Regimen.

Pub. Date : 2020 Sep

PMID : 32554434






1 Functional Relationships(s)
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1 Prolonged suppression of dehydroepiandrosterone (DHEA) concentrations observed in VCaP cells after abiraterone washout corroborated its protracted CYP17A1 engagement. Dehydroepiandrosterone cytochrome P450 family 17 subfamily A member 1 Homo sapiens