Title : Sigma-1 Receptor Agonist Amitriptyline Inhibits Store-Dependent Ca2+ Entry in Macrophages.

Pub. Date : 2019 Sep

PMID : 31768847






1 Functional Relationships(s)
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1 Using Fura-2AM microfluorimetry, we have shown for the first time that sigma-1 receptor agonist-tricyclic antidepressant amitriptyline-significantly inhibits store-dependent Ca2+ entry, induced by endoplasmic Ca2+-ATPase inhibitors thapsigargin and cyclopiazonic acid, in rat peritoneal macrophages. cyclopiazonic acid sigma non-opioid intracellular receptor 1 Rattus norvegicus