Title : Androgen Receptor Modulation Optimized for Response-Splice Variant: A Phase 3, Randomized Trial of Galeterone Versus Enzalutamide in Androgen Receptor Splice Variant-7-expressing Metastatic Castration-resistant Prostate Cancer.

Pub. Date : 2019 Dec

PMID : 31542304






1 Functional Relationships(s)
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Protein Name
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1 Galeterone inhibits CYP17 and AR, and induces AR protein degradation. 3-hydroxy-17-(1H-benzimidazole-1-yl)androsta-5,16-diene cytochrome P450 family 17 subfamily A member 1 Homo sapiens