Title : Design, synthesis and in vitro evaluation of 6-amide-2-aryl benzoxazole/benzimidazole derivatives against tumor cells by inhibiting VEGFR-2 kinase.

Pub. Date : 2019 Oct 1

PMID : 31252306






2 Functional Relationships(s)
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1 Design, synthesis and in vitro evaluation of 6-amide-2-aryl benzoxazole/benzimidazole derivatives against tumor cells by inhibiting VEGFR-2 kinase. benzimidazole kinase insert domain receptor Homo sapiens
2 A library of thirty-seven 6-amide-2-aryl benzoxazole/benzimidazole derivatives has been designed and synthesized based on the highly conserved active site of VEGFR-2. benzimidazole kinase insert domain receptor Homo sapiens