Title : Potent and selective caspase-2 inhibitor prevents MDM-2 cleavage in reversine-treated colon cancer cells.

Pub. Date : 2019 Dec

PMID : 30976094






3 Functional Relationships(s)
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1 Potent and selective caspase-2 inhibitor prevents MDM-2 cleavage in reversine-treated colon cancer cells. 2-(4-morpholinoanilino)-6-cyclohexylaminopurine caspase 2 Homo sapiens
2 Finally, we used the champion inhibitor (NH-23-C2) in reversine-treated HCT-116 colon cancer cells to selectively block caspase-2 activity and caspase-2-mediated MDM-2 cleavage. 2-(4-morpholinoanilino)-6-cyclohexylaminopurine caspase 2 Homo sapiens
3 Finally, we used the champion inhibitor (NH-23-C2) in reversine-treated HCT-116 colon cancer cells to selectively block caspase-2 activity and caspase-2-mediated MDM-2 cleavage. 2-(4-morpholinoanilino)-6-cyclohexylaminopurine caspase 2 Homo sapiens