Pub. Date : 2019 Feb
PMID : 30652318
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | In this study, hepatic uptake by recombinantly expressed monkey OATP1B1, OATP1B3 and OATP2B1 was investigated using three human OATP1B1 and OATP1B3 substrates (pitavastatin, pravastatin and rosuvastatin) and one OATP1B3 substrate (telmisartan), as the governmental drug interaction guidelines recommend, and seven reported clinical drugs. | Pravastatin | solute carrier organic anion transporter family member 1B1 | Homo sapiens |
2 | Consequently, pitavastatin, pravastatin and rosuvastatin were suggested to be substrates of recombinant monkey OATP1B1 and OATP1B3, and telmisartan was suggested to be a substrate of recombinant monkey OATP1B3, in a manner similar to human OATPs. | Pravastatin | solute carrier organic anion transporter family member 1B1 | Homo sapiens |