Title : Hypoxia-Activated Prodrugs of PERK Inhibitors.

Pub. Date : 2019 Apr 15

PMID : 30615821






1 Functional Relationships(s)
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1 We designed and prepared hypoxia-activated prodrugs of modified PERK inhibitors using a 2-nitroimidazole bioreductive trigger. azomycin eukaryotic translation initiation factor 2 alpha kinase 3 Homo sapiens