Pub. Date : 2019 Jan 15
PMID : 30553624
1 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Structural evolution of 37 produced the azide-containing cis-49a, which had good properties in three important respects: (1) selectivity for CYP1B1 over CYP1A1 and CYP1A2 (120-times and 150-times, respectively), (2) greater inhibitory potency of >2 times that of ANF, and (3) improved solubility. | Azides | cytochrome P450 family 1 subfamily A member 2 | Homo sapiens |