Title : Pharmacological characterization of JWX-A0108 as a novel type I positive allosteric modulator of α7 nAChR that can reverse acoustic gating deficits in a mouse prepulse inhibition model.

Pub. Date : 2019 Jun

PMID : 30333556






1 Functional Relationships(s)
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1 The alpha7 nicotinic acetylcholine receptor (alpha7 nAChR) is a ligand-gated Ca2+-permeable homopentameric ion channel implicated in cognition and neuropsychiatric disorders. Acetylcholine cholinergic receptor, nicotinic, alpha polypeptide 7 Mus musculus