Title : Antithrombotic P2Y12 receptor antagonists: recent developments in drug discovery.

Pub. Date : 2019 Jan

PMID : 30291899






1 Functional Relationships(s)
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1 Several different scaffolds have been identified as P2Y12 receptor antagonists, including irreversibly acting thienotetrahydropyridines (prodrugs), and reversible competitive antagonists, including adenine nucleotide analogs, piperazinyl-glutamate-quinolines, -pyridines, and -pyrimidines, and anthraquinone derivatives. Pyridines purinergic receptor P2Y12 Homo sapiens