Title : Screening for PPAR Non-Agonist Ligands Followed by Characterization of a Hit, AM-879, with Additional No-Adipogenic and cdk5-Mediated Phosphorylation Inhibition Properties.

Pub. Date : 2018

PMID : 29449830






2 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Peroxisome proliferator-activated receptor gamma (PPARgamma) is a member of a nuclear receptor superfamily and acts as a ligand-dependent transcription factor, playing key roles in maintenance of adipose tissue and in regulation of glucose and lipid homeostasis. Glucose peroxisome proliferator activated receptor gamma Homo sapiens
2 Peroxisome proliferator-activated receptor gamma (PPARgamma) is a member of a nuclear receptor superfamily and acts as a ligand-dependent transcription factor, playing key roles in maintenance of adipose tissue and in regulation of glucose and lipid homeostasis. Glucose peroxisome proliferator activated receptor gamma Homo sapiens